SCHEMBL25758432

SCHEMBL25758432

COc1ccc(NC(=O)c2ccc3ocnc3c2)cc1S(=O)(=O)Nc1c(C)cccc1C

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 9/20 0.49
KDM4E B2RXH2 5/20 0.49
GAA P10253 4/20 0.49
HTT P42858 3/20 0.49
POLB P06746 2/20 0.49
LMNA P02545 8/20 0.48
SMN1; SMN2 Q16637 4/20 0.48
HPGD P15428 2/20 0.48
NAMPT P43490 1/20 0.48
MEN1 O00255 7/20 0.47
KMT2A Q03164 7/20 0.47
ALDH1A1 P00352 5/20 0.47
ALOX12 P18054 1/20 0.47
CRHBP P24387 1/20 0.47
CRHR2 Q13324 1/20 0.47
HDAC1 Q13547 1/20 0.46
HDAC8 Q9BY41 1/20 0.46
HDAC6 Q9UBN7 1/20 0.46
CPT1A P50416 1/20 0.44
CPT1B Q92523 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23846415 0.93 MAPT (0.49) MAPTKDM4EGAAHTTPOLB
SCHEMBL23846996 0.85 MAPT (0.54) MAPTKDM4EGAAHTTPOLB
SCHEMBL23846444 0.83 NPC1 (0.58) MAPTKDM4EGAAHTTPOLB
SCHEMBL23846624 0.81 PRNP (0.56) MAPTKDM4EGAAHTTPOLB
SCHEMBL25754481 0.81 LMNA (0.47) MAPTKDM4EGAAHTTPOLB
SCHEMBL23846440 0.81 NPC1 (0.56) MAPTKDM4EGAAHTTPOLB
SCHEMBL23846477 0.81 NAMPT (0.46) MAPTKDM4EPOLBLMNASMN1; SMN2
SCHEMBL23846451 0.80 RAB9A (0.60) MAPTKDM4EGAAHTTPOLB
SCHEMBL25758408 0.80 MAPT (0.57) MAPTKDM4EGAAHTTPOLB
SCHEMBL23846398 0.80 NPC1 (0.52) MAPTKDM4EGAAHTTPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230174523-A1 BENZENESULFONAMIDE DERIVATIVES AS TRAP1 MODULATORS AND USES THEREOF AMATHUS THERAPEUTICS, INC. (US) 2023-06-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230174523-A1 BENZENESULFONAMIDE DERIVATIVES AS TRAP1 MODULATORS AND USES THEREOF TRAP1, PINK1, TP53BP1 MAPT 89/4885KDM4E 4448/4885GAA 1667/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.