SCHEMBL25787747

SCHEMBL25787747

NC(=O)c1cnc2c(c1)CCCN2

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NNMT P40261 7/20 1.00
KDM4E B2RXH2 1/20 0.42
MAPT P10636 1/20 0.42
CYP11B2 P19099 1/20 0.38
PIK3C3 Q8NEB9 1/20 0.38
CRBN Q96SW2 2/20 0.37
GRM5 P41594 1/20 0.36
CHRNB2 P17787 1/20 0.36
CHRNA4 P43681 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.35
ASIC3 Q9UHC3 1/20 0.35
OGA O60502 1/20 0.34
RPS6KA3 P51812 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25787741 0.90 NNMT (1.00) NNMTPIK3C3CRBNGRM5CHRNB2
SCHEMBL5306512 0.86 NNMT (0.75) NNMTKDM4EMAPTPIK3C3CRBN
SCHEMBL21782980 0.81 NNMT (0.68) NNMTKDM4EMAPTPIK3C3CRBN
SCHEMBL30968499 0.81 NNMT (0.68) NNMTKDM4EMAPTCYP11B2PIK3C3
SCHEMBL20722588 0.81 NNMT (0.68) NNMTKDM4EMAPTCYP11B2PIK3C3
SCHEMBL22226400 0.79 NNMT (0.64) NNMTKDM4ECYP11B2CRBNGRM5
SCHEMBL22226923 0.77 NNMT (0.63) NNMTKDM4E
SCHEMBL25787851 0.77 NNMT (0.62) NNMTGRM5CHRNB2CHRNA4
SCHEMBL25787975 0.77 NNMT (0.66) NNMTKDM4ECHRNB2CHRNA4SMN1; SMN2
SCHEMBL21772832 0.77 NNMT (0.62) NNMTKDM4EMAPTCYP11B2PIK3C3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110869363-B 5-membered and bicyclic heterocyclic amides as ROCK inhibitors 百时美施贵宝公司 2024-01-05 CN disclosed
WO-2023129512-A1 BICYCLIC INHIBITORS OF NICOTINAMIDE N-METHYLTRANSFERASE, COMPOSITIONS AND USES THEREOF PRESIDENT AND FELLOWS OF HARVARD COLLEGE (US) 2023-07-06 WO disclosed