SCHEMBL2579076

SCHEMBL2579076

Cc1nn(-c2ccccc2)nc1C(=O)N1CCc2onc(C(=O)NCc3cccnc3)c2C1

nearest known ligand 0.55

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.55
TP53 P04637 5/20 0.48
SMN1; SMN2 Q16637 4/20 0.46
KMT2A Q03164 2/20 0.46
LMNA P02545 2/20 0.46
NAMPT P43490 1/20 0.45
NPC1 O15118 1/20 0.45
HPGD P15428 1/20 0.45
RAB9A P51151 1/20 0.45
HDAC1 Q13547 1/20 0.45
ALDH1A1 P00352 1/20 0.44
TSHR P16473 2/20 0.44
HSP90AA1 P07900 1/20 0.44
KDM4E B2RXH2 1/20 0.43
HSD17B10 Q99714 1/20 0.43
ADORA2A P29274 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2580833 0.87 ALDH1A1 (0.53) GAASMN1; SMN2KMT2ALMNANPC1
SCHEMBL4265115 0.81 NPC1 (0.47) TP53SMN1; SMN2KMT2ALMNANPC1
SCHEMBL5530069 0.75 HDAC1 (0.42) TP53SMN1; SMN2KMT2ALMNANPC1
SCHEMBL15300384 0.74 MAPT (0.43) TP53SMN1; SMN2KMT2ALMNANPC1
SCHEMBL2587331 0.73 GAA (0.49) GAATP53SMN1; SMN2KMT2ALMNA
SCHEMBL13545878 0.72 GAA (1.00) GAATP53SMN1; SMN2KMT2ALMNA
SCHEMBL4263116 0.71 LMNA (0.56) GAASMN1; SMN2KMT2ALMNANPC1
SCHEMBL2588184 0.69 MAPT (0.63) GAASMN1; SMN2KMT2ALMNANPC1
SCHEMBL4263699 0.68 MAPT (0.60) GAASMN1; SMN2KMT2ALMNANAMPT
SCHEMBL2585124 0.66 LMNA (0.60) GAASMN1; SMN2KMT2ALMNANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8048879-B2 Substituted 4,5,6,7-tetrahydro-isoxazolo[4,5-c]pyridine compounds and use thereof for producing medicaments GRUENENTHAL GMBH (DE) 2011-11-01 US claimed
US-8048879-B2 Substituted 4,5,6,7-tetrahydro-isoxazolo[4,5-c]pyridine compounds and use thereof for producing medicaments GRUENENTHAL GMBH (DE) 2011-11-01 US disclosed