SCHEMBL257934

SCHEMBL257934

Cc1cc(F)cc(CI)c1

nearest known ligand 0.36

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ACHE P22303 2/20 0.36
RAPGEF4 Q8WZA2 2/20 0.33
IDO1 P14902 2/20 0.33
NR3C1 P04150 1/20 0.32
PGR P06401 1/20 0.32
NR3C2 P08235 1/20 0.32
NOS1 P29475 4/20 0.31
PGK1 P00558 1/20 0.31
PGK2 P07205 1/20 0.31
NOS3 P29474 2/20 0.30
NOS2 P35228 2/20 0.30
IDH1 O75874 1/20 0.30
RPS6KB1 P23443 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18475171 0.82 IDO1 (0.46) IDO1
SCHEMBL4957876 0.82 PGK1 (0.42) ACHEIDO1PGK1PGK2IDH1
SCHEMBL8340109 0.82 ALDH1A1 (0.40) ACHEPGK1PGK2IDH1
SCHEMBL14570491 0.80 ACHE (0.39) ACHERAPGEF4IDO1NR3C1PGR
SCHEMBL2662788 0.78 ACHE (0.37) ACHERAPGEF4IDO1NR3C1PGR
SCHEMBL7499745 0.78 ACHE (0.37) ACHERAPGEF4IDO1NR3C1PGR
SCHEMBL31614540 0.76 LOXL2 (0.42) ACHERAPGEF4IDO1NR3C1PGR
SCHEMBL16727024 0.76 ACHE (0.36) ACHERAPGEF4IDO1NR3C1PGR
SCHEMBL2924850 0.76 ACHE (0.36) ACHERAPGEF4IDO1NR3C1PGR
SCHEMBL4162524 0.76 LOXL2 (0.42) ACHERAPGEF4IDO1NR3C1PGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2399585-A1 Boronic acids and esters as inhibitors of fatty acid amide hydrolase Infinity Pharmaceuticals, Inc. (US) 2011-12-28 EP disclosed
EP-2073816-B1 BORONIC ACIDS AND ESTERS AS INHIBITORS OF FATTY ACID AMIDE HYDROLASE INFINITY PHARMACEUTICALS INC (US) 2011-09-14 EP disclosed
WO-2008063300-A2 BORONIC ACIDS AND ESTERS AS INHIBITORS OF FATTY ACID AMIDE HYDROLASE INFINITY PHARMACEUTICALS, INC. (US) 2008-05-29 WO disclosed