SCHEMBL25795155

SCHEMBL25795155

CC(C)(O)c1cc(C(F)(F)F)ccc1I

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.43
MEN1 O00255 3/20 0.41
KMT2A Q03164 3/20 0.41
KIF11 P52732 1/20 0.37
PDE2A O00408 5/20 0.37
CYP3A4 P08684 1/20 0.36
CYP2D6 P10635 1/20 0.36
AR P10275 1/20 0.35
ALOX15 P16050 1/20 0.35
TSHR P16473 1/20 0.35
MAPK1 P28482 1/20 0.35
HSD17B10 Q99714 1/20 0.35
CYP11B2 P19099 2/20 0.35
CYP11B1 P15538 1/20 0.35
PTPN5 P54829 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7630799 0.81 CES2 (0.50) CES2KIF11ARTSHRMAPK1
SCHEMBL17141574 0.78 MEN1 (0.44) CES2MEN1KMT2AKIF11PDE2A
SCHEMBL31618336 0.77 MAPT (0.43) CES2MEN1KMT2AKIF11PDE2A
SCHEMBL22507938 0.77 PGR (0.46) CES2MEN1KMT2AKIF11AR
SCHEMBL14016057 0.77 PDE2A (0.47) CES2MEN1KMT2APDE2ACYP3A4
SCHEMBL18358786 0.76 KIF11 (0.43) CES2MEN1KMT2AKIF11PDE2A
SCHEMBL24852666 0.74 ALDH1A1 (0.50) CES2MEN1KMT2APDE2ACYP3A4
SCHEMBL1529230 0.73 PDE2A (0.42) CES2MEN1KMT2AKIF11PDE2A
SCHEMBL31537454 0.73 PDE2A (0.42) CES2MEN1KMT2AKIF11PDE2A
SCHEMBL19544823 0.72 KIF11 (0.43) CES2MEN1KMT2AKIF11PDE2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023109912-A1 3, 4-DIHYDROISOQUINOLIN-1 (2H) -ONES DERIVATIVES AS STING ANTAGONISTS AND THE USE THEREOF BEIGENE, LTD. (KY) 2023-06-22 WO disclosed