SCHEMBL257994

SCHEMBL257994

COC(C)(C)C(C)(C)OBc1ccc(SCc2ccccc2)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC6A4 P31645 1/20 0.42
MAOA P21397 4/20 0.42
MAOB P27338 4/20 0.42
CYP3A4 P08684 2/20 0.37
PPARG P37231 2/20 0.37
PPARA Q07869 2/20 0.37
CYP2D6 P10635 2/20 0.37
CYP1A2 P05177 1/20 0.37
PRMT1 Q99873 1/20 0.37
APP P05067 1/20 0.37
LTA4H P09960 1/20 0.36
KDM4E B2RXH2 1/20 0.35
NPC1 O15118 1/20 0.35
ALDH1A1 P00352 1/20 0.35
TP53 P04637 1/20 0.35
GAA P10253 1/20 0.35
MAPT P10636 1/20 0.35
HPGD P15428 1/20 0.35
NFKB1 P19838 1/20 0.35
RAB9A P51151 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL257867 0.94 SLC6A4 (0.39) SLC6A4MAOAMAOBCYP3A4PPARG
SCHEMBL10089190 0.79 CES1 (0.32) ALDH1A1
SCHEMBL12330495 0.75 SLC6A4 (0.40) SLC6A4MAOAMAOBCYP3A4PPARG
SCHEMBL2433694 0.70 APP (0.69) SLC6A4MAOAMAOBPPARGPPARA
SCHEMBL27684871 0.70 EGFR (0.54) SLC6A4MAOAMAOBCYP3A4PPARG
SCHEMBL27285685 0.70 LTA4H (0.49) SLC6A4MAOAMAOBCYP3A4PPARG
SCHEMBL9972571 0.69 ACHE (0.34) ALDH1A1TDP1
SCHEMBL332623 0.68 MAOA (0.63) SLC6A4MAOAMAOBCYP3A4PPARG
SCHEMBL14232082 0.68 ENPP2 (0.34)
SCHEMBL10193348 0.68 CA1 (0.44) CYP3A4CYP1A2LTA4HKDM4ENPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2404607-A1 Boronic acids and esters as inhibitors of fatty acid amide hydrolase Infinity Pharmaceuticals, Inc. (US) 2012-01-11 EP disclosed
EP-2399585-A1 Boronic acids and esters as inhibitors of fatty acid amide hydrolase Infinity Pharmaceuticals, Inc. (US) 2011-12-28 EP disclosed
WO-2008063300-A2 BORONIC ACIDS AND ESTERS AS INHIBITORS OF FATTY ACID AMIDE HYDROLASE INFINITY PHARMACEUTICALS, INC. (US) 2008-05-29 WO disclosed