SCHEMBL25813723

SCHEMBL25813723

C[Si](C)(C)CCOCn1ccc2c(-c3cnn(CC4CCCC4)c3)ncnc21

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 2/20 0.38
PIK3CD O00329 2/20 0.34
PIK3CA P42336 2/20 0.34
JAK3 P52333 6/20 0.34
JAK2 O60674 4/20 0.34
SCN9A Q15858 1/20 0.33
ACACB O00763 1/20 0.32
DGAT1 O75907 1/20 0.32
JAK1 P23458 3/20 0.32
TYK2 P29597 1/20 0.32
BTK Q06187 1/20 0.32
PIM1 P11309 1/20 0.32
KDM5B Q9UGL1 1/20 0.32
SIGMAR1 Q99720 1/20 0.32
NPC1 O15118 1/20 0.31
RAB9A P51151 1/20 0.31
TTK P33981 1/20 0.31
PIK3CB P42338 1/20 0.31
PI4KA P42356 1/20 0.31
PIK3CG P48736 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21665752 0.89 JAK1 (0.34) LRRK2PIK3CDPIK3CAJAK3JAK2
SCHEMBL2383469 0.85 JAK2 (0.38) LRRK2PIK3CDPIK3CAJAK3JAK2
SCHEMBL6127068 0.84 JAK2 (0.35) LRRK2PIK3CDPIK3CAJAK3JAK2
SCHEMBL19601282 0.83 SIGMAR1 (0.43) LRRK2SCN9ADGAT1SIGMAR1
SCHEMBL2997635 0.83 JAK2 (0.36) LRRK2JAK3JAK2JAK1TYK2
SCHEMBL5133827 0.83 JAK2 (0.34) JAK3JAK2DGAT1JAK1TYK2
SCHEMBL5133826 0.83 TPH1 (0.35) LRRK2JAK3JAK2DGAT1JAK1
SCHEMBL22343499 0.81 LRRK2 (0.41) LRRK2PIK3CDPIK3CAJAK3JAK2
SCHEMBL100799 0.81 DGAT1 (0.35) JAK3JAK2DGAT1JAK1TYK2
SCHEMBL6127063 0.81 DGAT1 (0.34) DGAT1SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023125373-A1 METHOD FOR PREPARING RUXOLITINIB AND INTERMEDIATE THEREOF 江苏威凯尔医药科技有限公司 2023-07-06 WO disclosed