SCHEMBL25814190

SCHEMBL25814190

c1ccc2sc(CN3CCCC34CCNCC4)cc2c1

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.44
DRD4 P21917 1/20 0.44
DRD3 P35462 1/20 0.44
SLC6A2 P23975 1/20 0.42
CYP2A6 P11509 2/20 0.40
ASIC3 Q9UHC3 1/20 0.40
LOXL2 Q9Y4K0 1/20 0.40
FAAH O00519 2/20 0.39
MGLL Q99685 1/20 0.39
SIGMAR1 Q99720 7/20 0.39
MEN1 O00255 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
TSHR P16473 1/20 0.38
CYP2C19 P33261 1/20 0.38
THPO P40225 1/20 0.38
SLC6A3 Q01959 1/20 0.38
KMT2A Q03164 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25487489 0.84 FAAH (0.41) DRD2DRD4DRD3FAAHMGLL
SCHEMBL20566667 0.82 MGLL (0.57) SLC6A2FAAHMGLLMEN1CYP3A4
SCHEMBL20778554 0.73 MGLL (0.57) MGLL
SCHEMBL19582597 0.69 MAPT (0.42) SLC6A2SIGMAR1MEN1CYP2D6TSHR
SCHEMBL10238584 0.69 FAAH (0.56) DRD2DRD4DRD3SLC6A2CYP2A6
SCHEMBL15084320 0.69 DRD2 (0.54) DRD2DRD4DRD3CYP2A6ASIC3
SCHEMBL1556809 0.66 CYP2D6 (0.50) SIGMAR1MEN1CYP3A4CYP2D6TSHR
SCHEMBL807399 0.66 DRD2 (0.47) DRD2DRD4DRD3SLC6A2CYP2A6
SCHEMBL19603152 0.65 SIGMAR1 (0.49) SLC6A2SIGMAR1MEN1KMT2A
SCHEMBL13499604 0.64 FAAH (0.57) DRD2DRD4DRD3SLC6A2CYP2A6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3675847-B1 SPIROCYCLE COMPOUNDS AND METHODS OF MAKING AND USING SAME H LUNDBECK AS (DK) 2023-07-12 EP disclosed