SCHEMBL25814826

SCHEMBL25814826

CC(C)(N)c1cccc(C#N)c1F

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.36
SLC22A12 Q96S37 1/20 0.35
NOTUM Q6P988 1/20 0.35
LRRK2 Q5S007 1/20 0.35
AR P10275 8/20 0.34
MAP2K1 Q02750 1/20 0.34
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
PDK1 Q15118 1/20 0.33
PDK2 Q15119 1/20 0.33
PDK3 Q15120 1/20 0.33
PDK4 Q16654 1/20 0.33
ALDH1A1 P00352 1/20 0.33
HTT P42858 1/20 0.33
PGR P06401 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL19532870 0.85 CA2 (0.40) TSHRSLC22A12NOTUMARPDK1
SCHEMBL6804271 0.81 GABRA1 (0.40) TSHRSLC22A12NOTUMARPDK1
SCHEMBL151808 0.80 TSHR (0.46) TSHRSLC22A12ARMAP2K1CYP1A2
SCHEMBL2003310 0.79 AR (0.46) SLC22A12ARPGR
SCHEMBL1533157 0.75 TSHR (0.46) TSHRNOTUMLRRK2MAP2K1CYP1A2
SCHEMBL23886265 0.74 HSD11B1 (0.37)
SCHEMBL30018006 0.74 HSD11B1 (0.37)
SCHEMBL30018336 0.72 KIF11 (0.45) TSHRCYP1A2CYP3A4PDK2ALDH1A1
Hydrochloric Acid SCHEMBL29168009 0.72 HTR2C (0.37)
SCHEMBL23886233 0.72 KIF11 (0.45) TSHRCYP1A2CYP3A4PDK2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023125737-A1 HETEROCYCLIC COMPOUNDS AND USE THEREOF SILEXON AI TECHNOLOGY CO., LTD. (CN) 2023-07-06 WO disclosed