SCHEMBL2581642

SCHEMBL2581642

N#Cc1c(C(=O)O)cccc1-n1ccc2ccccc21

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.40
ALB P02768 1/20 0.40
HSP90AA1 P07900 2/20 0.39
TRAP1 Q12931 2/20 0.39
HSP90AB1 P08238 1/20 0.39
HSP90B1 P14625 1/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
POLB P06746 1/20 0.39
APEX1 P27695 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
NOTUM Q6P988 1/20 0.38
NR4A1 P22736 1/20 0.38
NR4A2 P43354 1/20 0.38
NR4A3 Q92570 1/20 0.38
ALOX15 P16050 1/20 0.38
CDC25B P30305 1/20 0.38
HSD17B10 Q99714 1/20 0.37
KMT2A Q03164 2/20 0.37
TSHR P16473 1/20 0.37
RAB9A P51151 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28436731 0.82 L3MBTL1 (0.56) ALDH1A1HSP90AA1TRAP1HSP90AB1HSP90B1
SCHEMBL16720449 0.80 PTPN22 (0.38) ALDH1A1HSP90AA1TRAP1HSP90AB1HSP90B1
SCHEMBL484192 0.79 MYC (0.46) ALDH1A1HSP90AA1TRAP1HSP90AB1HSP90B1
SCHEMBL2581647 0.78 ALB (0.40) ALBL3MBTL1POLBNOTUMNR4A1
SCHEMBL8926318 0.73 HTR3A (0.45) ALDH1A1L3MBTL1POLBAPEX1TDP1
SCHEMBL152899 0.73 HSP90AA1 (0.50) ALDH1A1HSP90AA1TRAP1HSP90AB1HSP90B1
SCHEMBL154462 0.72 NOTUM (0.50) ALDH1A1HSP90AA1TRAP1HSP90AB1HSP90B1
SCHEMBL30637639 0.72 NPC1 (0.46) ALDH1A1HSP90AA1TRAP1HSP90AB1HSP90B1
SCHEMBL30928942 0.72 NPC1 (0.46) ALDH1A1HSP90AA1TRAP1HSP90AB1HSP90B1
SCHEMBL8610906 0.72 NPC1 (0.46) ALDH1A1HSP90AA1TRAP1HSP90AB1HSP90B1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2383573-A1 SCREENING METHOD FOR SUBSTANCE USEFUL AS AGENT FOR TREATING PROSTATE CANCER Astellas Pharma Inc. (JP) 2011-11-02 EP disclosed