SCHEMBL8926318

SCHEMBL8926318

N#Cc1ccccc1-n1ccc2c(C(=O)O)cccc21

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 1/20 0.45
HTR7 P34969 1/20 0.43
ALDH1A1 P00352 3/20 0.43
KMT2A Q03164 1/20 0.42
NOTUM Q6P988 1/20 0.41
GALR3 O60755 1/20 0.41
RAB9A P51151 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.40
XIAP P98170 1/20 0.40
SCN9A Q15858 2/20 0.39
TSHR P16473 2/20 0.39
POLB P06746 1/20 0.39
APEX1 P27695 1/20 0.39
TDP1 Q9NUW8 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9428481 0.77 TSHR (0.46) HTR3AHTR7ALDH1A1KMT2ASMN1; SMN2
SCHEMBL9429028 0.77 HTR7 (0.47) HTR3AHTR7ALDH1A1KMT2AGALR3
SCHEMBL15565198 0.77 HTR7 (0.40) HTR3AHTR7ALDH1A1KMT2ASMN1; SMN2
SCHEMBL17176324 0.77 ALDH1A1 (0.63) HTR3AHTR7ALDH1A1KMT2AGALR3
SCHEMBL19643369 0.76 NOTUM (0.53) ALDH1A1NOTUMPOLBAPEX1TDP1
SCHEMBL9445884 0.75 NOTUM (0.44) HTR3AHTR7KMT2ANOTUMTSHR
SCHEMBL9343076 0.74 XIAP (0.44) HTR3AHTR7ALDH1A1KMT2AGALR3
SCHEMBL17170720 0.74 TSHR (0.67) HTR3AHTR7ALDH1A1KMT2AGALR3
SCHEMBL9429365 0.73 FABP4 (0.56) ALDH1A1KMT2ANOTUMTSHRPOLB
SCHEMBL2581642 0.73 ALDH1A1 (0.40) ALDH1A1KMT2ANOTUMRAB9ATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5616591-A Indole- and benzimidazole-substituted quinoline derivatives E.R. SQUIBB & SONS, INC. (US) 1997-04-01 US disclosed
US-5374615-A Treating hypertension and congestive heart failure, preventing cardiac hypertrophy E. R. SQUIBB & SONS, INC. (US) 1994-12-20 US disclosed
US-5236916-A Oxadiazinone substituted indole and benzimidazole derivatives E. R. SQUIBB & SONS, INC. (US) 1993-08-17 US disclosed
US-5208235-A Phosphonic or phosphinic acid derivatives as inhibitors of angiotnesin II for cardiovascular disorders and hypotensives E. R. SQUIBB & SONS, INC. (US) 1993-05-04 US disclosed
EP-0488532-A1 Indole- and benzimidazole-substituted imidazole and benzimidazole derivatives E.R. Squibb & Sons, Inc. (US) 1992-06-03 EP disclosed