SCHEMBL25819366

SCHEMBL25819366

COCCc1nc2cnc3ccsc3c2n1CC1CCN(C(=O)OC(C)(C)C)CC1

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 5/20 0.43
ADORA2B P29275 5/20 0.43
FEN1 P39748 1/20 0.39
USP7 Q93009 1/20 0.39
PIK3CA P42336 1/20 0.39
PRKDC P78527 1/20 0.39
SYK P43405 1/20 0.39
KDM4E B2RXH2 1/20 0.38
PKM P14618 1/20 0.38
GPR119 Q8TDV5 5/20 0.38
ADORA3 P0DMS8 1/20 0.38
BACE1 P56817 1/20 0.37
LMNA P02545 1/20 0.37
RORC P51449 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31270644 0.90 ADORA2A (0.41) ADORA2AADORA2BFEN1USP7PIK3CA
SCHEMBL25256593 0.90 ADORA2A (0.41) ADORA2AADORA2BFEN1USP7PIK3CA
SCHEMBL31270561 0.85 ADORA2A (0.38) ADORA2AADORA2BFEN1PIK3CAPRKDC
SCHEMBL25300972 0.85 ADORA2A (0.38) ADORA2AADORA2BFEN1PIK3CAPRKDC
SCHEMBL25260626 0.83 ADORA2A (0.42) ADORA2AADORA2BFEN1SYKKDM4E
SCHEMBL31270757 0.83 ADORA2A (0.42) ADORA2AADORA2BFEN1SYKKDM4E
SCHEMBL25262168 0.77 ADORA2B (0.41) ADORA2BPIK3CAPRKDCGPR119LMNA
SCHEMBL31270748 0.77 ADORA2B (0.41) ADORA2BPIK3CAPRKDCGPR119LMNA
SCHEMBL31270623 0.76 GLS (0.39) PIK3CAPRKDCGPR119LMNARORC
SCHEMBL25819006 0.76 GLS (0.39) PIK3CAPRKDCGPR119LMNARORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260055119-A9 TRICYCLIC COMPOUND, METHOD FOR PREPARING SAME, AND USE THEREOF SICHUAN KELUN BIOTECH BIOPHARMACEUTICAL CO LTD (CN) 2026-02-26 US disclosed
US-20250257071-A9 TRICYCLIC COMPOUND, METHOD FOR PREPARING SAME, AND USE THEREOF SICHUAN KELUN-BIOTECH BIOPHARMACEUTICAL CO., LTD. (CN) 2025-08-14 US disclosed
US-20250002502-A1 TRICYCLIC COMPOUND, METHOD FOR PREPARING SAME, AND USE THEREOF SICHUAN KELUN BIOTECH BIOPHARMACEUTICAL CO LTD (CN) 2025-01-02 US disclosed
EP-4458830-A1 TRICYCLIC COMPOUND, METHOD FOR PREPARING SAME, AND USE THEREOF Sichuan Kelun-Biotech Biopharmaceutical Co., Ltd. (CN) 2024-11-06 EP disclosed
CN-118201933-A Tri-fused ring compounds, preparation method and application thereof 四川科伦博泰生物医药股份有限公司 2024-06-14 CN disclosed
WO-2023125121-A1 TRICYCLIC COMPOUND, METHOD FOR PREPARING SAME, AND USE THEREOF 四川科伦博泰生物医药股份有限公司 2023-07-06 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20250257071-A9 TRICYCLIC COMPOUND, METHOD FOR PREPARING SAME, AND USE THEREOF CYP11B2, CYP11B1, CYP3A5 ADORA2A 1834/4885ADORA2B 1831/4885FEN1 4208/4885
US-20260055119-A9 TRICYCLIC COMPOUND, METHOD FOR PREPARING SAME, AND USE THEREOF CYP11B1, CYP11B2, CYP2D6 ADORA2A 2615/4885ADORA2B 2385/4885FEN1 3630/4885
US-20250002502-A1 TRICYCLIC COMPOUND, METHOD FOR PREPARING SAME, AND USE THEREOF CYP11B2, CYP11B1, CYP3A5 ADORA2A 1834/4885ADORA2B 1831/4885FEN1 4208/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.