SCHEMBL2582155

SCHEMBL2582155

Oc1cccc(Oc2ccccn2)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TLR4 O00206 1/20 0.50
TLR2 O60603 1/20 0.50
MGLL Q99685 1/20 0.50
GRM5 P41594 1/20 0.48
FFAR4 Q5NUL3 1/20 0.47
MAP4K4 O95819 1/20 0.45
KDM4E B2RXH2 1/20 0.44
RET P07949 1/20 0.43
KIF5B P33176 1/20 0.43
KDR P35968 1/20 0.43
IP6K1 Q92551 1/20 0.43
IP6K3 Q96PC2 1/20 0.43
IP6K2 Q9UHH9 1/20 0.43
PPARG P37231 1/20 0.42
RAB9A P51151 1/20 0.41
HRH3 Q9Y5N1 1/20 0.41
CYP3A4 P08684 1/20 0.41
PTGS2 P35354 2/20 0.40
MBD2 Q9UBB5 1/20 0.40
DRD1 P21728 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30843232 1.00 TLR4 (0.50) TLR4TLR2MGLLGRM5FFAR4
SCHEMBL29612417 0.87 TLR4 (0.56) TLR4TLR2GRM5FFAR4MAP4K4
SCHEMBL12129555 0.87 TLR4 (0.56) TLR4TLR2GRM5FFAR4MAP4K4
SCHEMBL15602369 0.85 TLR4 (0.55) TLR4TLR2GRM5FFAR4MAP4K4
SCHEMBL5686998 0.83 SCN7A (0.47) TLR4TLR2MGLLKDM4EPPARG
SCHEMBL15387423 0.82 HRH3 (0.44) TLR4TLR2MGLLGRM5FFAR4
SCHEMBL3334396 0.82 ESR2 (0.53) TLR4TLR2MGLLGRM5MAP4K4
SCHEMBL5109000 0.81 MAP4K4 (0.57) TLR4TLR2GRM5FFAR4MAP4K4
SCHEMBL12168388 0.81 F2 (0.53) KDM4ERETKIF5BKDRRAB9A
SCHEMBL6091732 0.81 CHRNB2 (0.51) MGLLAPP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 130 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-55108851-A None JP disclosed
US-20260035398-A1 TETRADENTATE AND OCTAHEDRAL METAL COMPLEXES CONTAINING NAPHTHYRIDINOCARBAZOLE AND ITS ANALOGUES UNIV ARIZONA STATE (US) 2026-02-05 US disclosed
US-12457894-B2 Organometallic compound and organic light-emitting device including the same SAMSUNG DISPLAY CO., LTD. (KR) 2025-10-28 US disclosed
US-12312366-B2 Tetradentate and octahedral metal complexes containing naphthyridinocarbazole and its analogues ARIZONA BOARD OF REGENTS ON BEHALF OF ARIZONA STATE UNIVERSITY (US) 2025-05-27 US disclosed
EP-4185858-B1 COMPOSITIONS, SYSTEMS AND METHODS FOR BIOLOGICAL ANALYSIS USING DYES LIFE TECHNOLOGIES CORP (US) 2025-05-21 EP disclosed
US-11998538-B2 Piperidine urea derivatives as soluble epoxide hydrolase inhibitors NEUROPN THERAPEUTICS (US) 2024-06-04 US disclosed
US-11998538-B2 Piperidine urea derivatives as soluble epoxide hydrolase inhibitors NEUROPN THERAPEUTICS (US) 2024-06-04 US disclosed
CN-110272456-B Organometallic compound and organic light emitting device including the same 三星显示有限公司 2024-04-05 CN disclosed
US-20240060117-A1 ENERGY TRANSFER DYE CONJUGATES FOR USE IN BIOLOGICAL ASSAYS Life Technologies Corporation 2024-02-22 US disclosed
EP-4306521-A1 CENTRAL CHIRALITY INDUCED SPIRO CHIRAL TETRADENTATE CYCLOMETALATED PLATINUM (II) AND PALLADIUM (II) COMPLEX-BASED CIRCULARLY POLARIZED LUMINESCENCE MATERIAL AND APPLICATION THEREOF Zhejiang University of Technology (CN) 2024-01-17 EP disclosed
WO-2011137431-A2 SYNTHESIS OF FOUR COORDINATED GOLD COMPLEXES AND THEIR APPLICATIONS IN LIGHT EMITTING DEVICES THEREOF ARIZONA BOARD OF REGENTS FOR AND ON BEHALF OF ARIZONA STATE UNIVERSITY (US) 2011-11-03 WO disclosed
WO-2011137431-A2 SYNTHESIS OF FOUR COORDINATED GOLD COMPLEXES AND THEIR APPLICATIONS IN LIGHT EMITTING DEVICES THEREOF ARIZONA BOARD OF REGENTS FOR AND ON BEHALF OF ARIZONA STATE UNIVERSITY (US) 2011-11-03 WO disclosed
WO-2011137429-A2 SYNTHESIS OF FOUR COORDINATED PALLADIUM COMPLEXES AND THEIR APPLICATIONS IN LIGHT EMITTING DEVICES THEREOF ARIZONA BOARD OF REGENTS ACTING FOR AND ON BEHALF OF ARIZONA STATE UNIVERSITY (US) 2011-11-03 WO disclosed
WO-2011137429-A2 SYNTHESIS OF FOUR COORDINATED PALLADIUM COMPLEXES AND THEIR APPLICATIONS IN LIGHT EMITTING DEVICES THEREOF ARIZONA BOARD OF REGENTS ACTING FOR AND ON BEHALF OF ARIZONA STATE UNIVERSITY (US) 2011-11-03 WO disclosed
WO-2010118026-A2 SYNTHESIS OF FOUR COORDINATED PLATINUM COMPLEXES AND THEIR APPLICATIONS IN LIGHT EMITTING DEVICES THEREOF ARIZONA BOARD OF REGENTS ACTING FOR AND ON BEHALF OF ARIZONA STATE UNIVERSITY (US) 2010-10-14 WO disclosed
US-7781074-B2 Organic electroluminescent element FUJIFILM CORPORATION (JP) 2010-08-24 US disclosed
US-7781074-B2 Organic electroluminescent element FUJIFILM CORPORATION (JP) 2010-08-24 US disclosed
US-4455427-A THROMBOXANE INHIBITORS THE UPJOHN COMPANY (US) 1984-06-19 US disclosed
EP-0069521-A2 Pyridinyl and imidazolyl derivatives of benzofurans and benzothiophenes THE UPJOHN COMPANY (US) 1983-01-12 EP disclosed
JP-S55108851-A DERIVATIVE OF CARBAMIC ACID ESTER MITSUI TOATSU CHEM INC 1980-08-21 JP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20260035398-A1 TETRADENTATE AND OCTAHEDRAL METAL COMPLEXES CONTAINING NAPHTHYRIDINOCARBAZOLE AND ITS ANALOGUES LBR, SCO2, RAD54L TLR4 2997/4885TLR2 3466/4885MGLL 1684/4885
US-12457894-B2 Organometallic compound and organic light-emitting device including the same CRY1, OCIAD1, ORC3 TLR4 4148/4885TLR2 4110/4885MGLL 1473/4885
US-12312366-B2 Tetradentate and octahedral metal complexes containing naphthyridinocarbazole and its analogues PAICS, DNTT, PNPO TLR4 3043/4885TLR2 4185/4885MGLL 3447/4885
US-11998538-B2 Piperidine urea derivatives as soluble epoxide hydrolase inhibitors EPHX1, EPHX2, HPGDS TLR4 4240/4885TLR2 4714/4885MGLL 731/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.