SCHEMBL2582687

SCHEMBL2582687

Cc1c(Cc2ccc(-c3cn[nH]c3)cc2)c(OC(F)F)nc2c(Cl)ccc([O])c12

nearest known ligand 0.35

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 10/20 0.35
ROCK1 Q13464 1/20 0.35
KCNH2 Q12809 2/20 0.34
GRIN2B Q13224 1/20 0.34
AKT1 P31749 4/20 0.33
PRKD3 O94806 1/20 0.32
PRKCG P05129 1/20 0.32
PRKCB P05771 1/20 0.32
BRAF P15056 1/20 0.32
PRKCA P17252 1/20 0.32
PRKCH P24723 1/20 0.32
PRKCI P41743 1/20 0.32
PRKCE Q02156 1/20 0.32
PRKCQ Q04759 1/20 0.32
PRKCZ Q05513 1/20 0.32
PRKCD Q05655 1/20 0.32
PRKD1 Q15139 1/20 0.32
AKT2 P31751 4/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2581492 0.85 KCNH2 (0.34) KCNH2GRIN2B
SCHEMBL2573522 0.85 PTGDR2 (0.38) ROCK2ROCK1
SCHEMBL533986 0.82 AR (0.36)
SCHEMBL2580572 0.81 TGFBR1 (0.32)
SCHEMBL2579240 0.78 PTGDR2 (0.34)
SCHEMBL2574953 0.76 PTGDR2 (0.44)
SCHEMBL2574519 0.75 USP1 (0.33)
SCHEMBL2570608 0.74 KCNH2 (0.36) KCNH2
SCHEMBL2580081 0.74 USP1 (0.32) GRIN2B
SCHEMBL2571385 0.72 PTGDR2 (0.41) KCNH2GRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2139881-B1 QUINOLINES AND THEIR THERAPEUTIC USE PULMAGEN THERAPEUTICS ASTHMA LTD (GB) 2011-11-09 EP claimed