SCHEMBL25832502

SCHEMBL25832502

CCCCOc1cc2c(cc1C)C(=NCc1ccccc1)CC1(CCCCC1)C2

nearest known ligand 0.34

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.34
RARB P10826 1/20 0.33
NPSR1 Q6W5P4 1/20 0.32
RXRA P19793 1/20 0.32
WDR5 P61964 1/20 0.31
GRIN1 Q05586 1/20 0.30
GRIN2A Q12879 1/20 0.30
GRIN2B Q13224 1/20 0.30
SLC6A5 Q9Y345 1/20 0.30
LMNA P02545 1/20 0.30
TP53 P04637 1/20 0.30
MAPT P10636 1/20 0.30
C5AR1 P21730 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25832276 0.82 NPSR1 (0.34) RARBNPSR1RXRAWDR5LMNA
SCHEMBL25832499 0.77 RARB (0.36) THRBRARBNPSR1SLC6A5LMNA
SCHEMBL25832189 0.77 ACAT2 (0.39) NPSR1MAPT
SCHEMBL25832488 0.64 CNR2 (0.38) THRBRARBRXRAWDR5
SCHEMBL22898902 0.64 REN (0.36)
SCHEMBL9701936 0.64 MAPK1 (0.51) RARBMAPTC5AR1
SCHEMBL12434156 0.59 ESR1 (0.49) THRBRARBNPSR1WDR5LMNA
SCHEMBL16351328 0.59 TLR8 (0.55) MAPT
SCHEMBL25832275 0.59 RARB (0.36) THRBRARBNPSR1RXRALMNA
SCHEMBL27501527 0.58 RARB (0.56) THRBRARBLMNAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11702427-B2 Substituted 2-pyridone tricyclic compounds, analogues thereof, and methods using same ARBUTUS BIOPHARMA CORPORATION (CA) 2023-07-18 US disclosed
US-9676760-B2 Fused heterocyclic compounds as ion channel modulators GILEAD SCIENCES, INC. (US) 2017-06-13 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11702427-B2 Substituted 2-pyridone tricyclic compounds, analogues thereof, and methods using same HAVCR2, HPD, CYP24A1 THRB 1401/4885RARB 1652/4885NPSR1 3509/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.