SCHEMBL25838310

SCHEMBL25838310

COc1cc(N2CCc3cc(C)cc([C@@H]4CCCN4)c3C2)ccn1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
CYP17A1 P05093 3/20 0.34
CHRM4 P08173 2/20 0.34
CHRM2 P08172 1/20 0.34
PIK3CD O00329 2/20 0.34
EED O75530 1/20 0.34
SMARCA2 P51531 2/20 0.33
SMARCA4 P51532 2/20 0.33
CHRNB2 P17787 1/20 0.33
CHRNB4 P30926 1/20 0.33
CHRNA4 P43681 1/20 0.33
CHRNA2 Q15822 1/20 0.33
PSEN1 P49768 3/20 0.33
PSEN2 P49810 3/20 0.33
APH1B Q8WW43 3/20 0.33
NCSTN Q92542 3/20 0.33
APH1A Q96BI3 3/20 0.33
PSENEN Q9NZ42 3/20 0.33
OPRM1 P35372 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25838311 0.85 CHRM4 (0.35) CYP17A1CHRM4CHRM2EEDPSEN1
SCHEMBL30068955 0.82 PIK3CG (0.34) PIK3CD
SCHEMBL25256216 0.82 PIK3CG (0.34) PIK3CD
SCHEMBL25302991 0.82 PIK3CG (0.34) PIK3CD
SCHEMBL25838493 0.80 CHRNB2 (0.33) MEN1KMT2ACHRNB2CHRNB4CHRNA4
SCHEMBL25838278 0.78 TLR9 (0.34) EED
SCHEMBL25838282 0.78 HSD17B10 (0.31)
SCHEMBL30491189 0.77 AOC3 (0.32) MEN1KMT2AEED
SCHEMBL30491458 0.74 EED (0.40) MEN1KMT2AEEDCHRNB2CHRNA4
SCHEMBL25838296 0.74 PDE4B (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023131122-A1 FUSED RING-SUBSTITUTED SIX-MEMBERED HETEROCYCLIC COMPOUND, AND PREPARATION METHOD THEREFOR AND USE THEREOF 劲方医药科技(上海)有限公司 2023-07-13 WO disclosed