SCHEMBL2583837

SCHEMBL2583837

CCC(I)(c1ccccc1)c1ccccc1

nearest known ligand 0.52

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
KCNN4 O15554 4/20 0.44
TAAR1 Q96RJ0 1/20 0.41
MAPK1 P28482 1/20 0.39
KIF11 P52732 4/20 0.38
TSHR P16473 2/20 0.38
ALDH1A1 P00352 2/20 0.38
TP53 P04637 1/20 0.38
CYP2C19 P33261 1/20 0.37
HIF1A Q16665 1/20 0.37
ALOX15 P16050 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7339642 0.80 KCNN4 (0.41) KCNN4TAAR1MAPK1KIF11TSHR
Iodide SCHEMBL28547565 0.78 KCNN4 (0.40) KCNN4TAAR1MAPK1KIF11TSHR
SCHEMBL20752446 0.78 TAAR1 (0.41) KCNN4TAAR1MAPK1ALDH1A1TP53
SCHEMBL1971090 0.78 KCNN4 (0.48) KCNN4TAAR1MAPK1KIF11TSHR
SCHEMBL540402 0.77 KCNN4 (0.43) KCNN4TAAR1MAPK1KIF11TSHR
SCHEMBL6678725 0.77 TAAR1 (0.44) KCNN4TAAR1MAPK1TSHRALDH1A1
SCHEMBL6682491 0.76 KCNN4 (0.46) KCNN4TAAR1MAPK1TSHRALDH1A1
SCHEMBL14743401 0.75 KIF11 (0.37) MAPK1KIF11TSHRALDH1A1CYP2C19
SCHEMBL2208547 0.75 CYP2C19 (0.41) KCNN4TAAR1ALDH1A1CYP2C19HIF1A
SCHEMBL21577161 0.73 SIGMAR1 (0.40) MAPK1KIF11TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011137331-A2 4-FLUORO-4-ARYLPIPERDIN-1-YL DERIVATIVES AS MU OPIOID FUNCTION MODERATORS KINENTIA BIOSCIENCES LLC (US) 2011-11-03 WO disclosed
EP-0771196-A4 EXCITATORY AMINO ACID RECEPTOR ANTAGONISTS LILLY CO ELI (US) 1997-09-03 EP disclosed
EP-0771196-A1 EXCITATORY AMINO ACID RECEPTOR ANTAGONISTS ELI LILLY AND COMPANY (US) 1997-05-07 EP disclosed
WO-1996007405-A1 EXCITATORY AMINO ACID RECEPTOR ANTAGONISTS ELI LILLY AND COMPANY (US) 1996-03-14 WO disclosed
WO-1996005828-A1 PYRROLIDINYL DI-CARBOXYLIC ACID DERIVATIVES AS METABOTROPIC GLUTAMATE RECEPTOR ANTAGONISTS ELI LILLY AND COMPANY (US) 1996-02-29 WO disclosed