SCHEMBL2585043

SCHEMBL2585043

Cc1c(-c2ccoc2)n[nH]c1B(O)O

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TTK P33981 1/20 0.40
LRRK2 Q5S007 15/20 0.38
NTRK1 P04629 1/20 0.36
PIM1 P11309 1/20 0.35
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
HPGD P15428 1/20 0.33
HTT P42858 1/20 0.33
HSD17B10 Q99714 1/20 0.33
ADORA2A P29274 1/20 0.33
ADORA1 P30542 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1701209 0.72 HSP90AA1 (0.48) KDM4EALDH1A1HPGDHTTHSD17B10
SCHEMBL1701249 0.67 KDM4E (0.41) KDM4EALDH1A1HPGDHSD17B10ADORA2A
SCHEMBL1701438 0.66 HTR7 (0.41) PIM1KDM4EHPGD
SCHEMBL29643870 0.64 NTRK1 (0.40) TTKLRRK2NTRK1PIM1ADORA2A
SCHEMBL22890550 0.64 NTRK1 (0.40) TTKLRRK2NTRK1PIM1ADORA2A
SCHEMBL3256526 0.64 IDO1 (0.61) TTKLRRK2NTRK1PIM1KDM4E
SCHEMBL29771525 0.64 IDO1 (0.61) TTKLRRK2NTRK1PIM1KDM4E
SCHEMBL20919925 0.63 DYRK1A (0.46)
SCHEMBL12066975 0.62 TTK (0.36) TTKLRRK2NTRK1PIM1KDM4E
SCHEMBL3775393 0.61 TTK (0.66) TTKLRRK2NTRK1PIM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2563759-A2 COMPOUNDS THAT MODULATE INTRACELLULAR CALCIUM Calcimedica, Inc. (US) 2013-03-06 EP disclosed
WO-2011139765-A2 COMPOUNDS THAT MODULATE INTRACELLULAR CALCIUM CALCIMEDICA, INC. (US) 2011-11-10 WO disclosed