SCHEMBL25852175

SCHEMBL25852175

C=Cc1cc(C)c(Cl)c(Cl)c1

nearest known ligand 0.36

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 2/20 0.36
CHRM1 P11229 1/20 0.36
ALOX15 P16050 1/20 0.36
MAOA P21397 1/20 0.36
TBXA2R P21731 1/20 0.36
ADRA1A P35348 1/20 0.36
HTR2B P41595 1/20 0.36
TP53 P04637 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
RAPGEF4 Q8WZA2 1/20 0.35
SIRT1 Q96EB6 1/20 0.33
ALDH1A1 P00352 2/20 0.32
PTGS1 P23219 2/20 0.31
PTGS2 P35354 2/20 0.31
ALOX5 P09917 1/20 0.31
CD44 P16070 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6512393 0.88 CYP3A4 (0.46) CYP3A4CHRM1ALOX15MAOATBXA2R
SCHEMBL1122678 0.83 ALDH1A1 (0.45) CYP3A4TP53TDP1ALDH1A1
SCHEMBL10899149 0.82 TP53 (0.35) TP53TDP1ALDH1A1PTGS1PTGS2
SCHEMBL18611534 0.78 TP53 (0.33) TP53TDP1PTGS1PTGS2
SCHEMBL25142209 0.78 PTGS1 (0.49) CYP3A4ALOX15SIRT1ALDH1A1PTGS1
SCHEMBL15107889 0.78 TP53 (0.39) TP53TDP1ALDH1A1
SCHEMBL23464454 0.77 ALDH1A1 (0.46) CYP3A4CHRM1ALOX15MAOATBXA2R
SCHEMBL20144645 0.76 RAPGEF4 (0.38) CYP3A4CHRM1ALOX15MAOATBXA2R
SCHEMBL578860 0.73 TDP1 (0.45) CYP3A4TP53TDP1ALDH1A1PTGS1
SCHEMBL1122511 0.73 CYP3A4 (0.46) CYP3A4TP53TDP1RAPGEF4ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023135233-A1 AZAINDOLE DERIVATIVES AND THEIR USE AS ERK KINASE INHIBITORS AGV DISCOVERY (FR) 2023-07-20 WO disclosed