SCHEMBL25856428

SCHEMBL25856428

Cc1cc(N)nnc1-c1ccc(C#CBr)cc1O

nearest known ligand 0.36

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
NLRP3 Q96P20 6/20 0.36
IL1B P01584 3/20 0.34
TNF P01375 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25859518 0.87 NLRP3 (0.37) NLRP3IL1BTNF
SCHEMBL25856432 0.83 NLRP3 (0.38) NLRP3IL1BTNF
SCHEMBL25519380 0.83 NLRP3 (0.50) NLRP3IL1B
SCHEMBL25859262 0.82 IL1B (0.43) NLRP3IL1BTNF
SCHEMBL25856423 0.79 NLRP3 (0.30) NLRP3
SCHEMBL25861298 0.74 KDM4E (0.41)
SCHEMBL26773007 0.72 TRPA1 (0.44) IL1B
SCHEMBL30833885 0.72 IL1B (0.72) NLRP3IL1BTNF
SCHEMBL25857850 0.71 NLRP3 (0.42) NLRP3IL1BTNF
SCHEMBL24575631 0.71 SIRT3 (0.37) IL1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023131277-A1 NLRP3 INFLAMMASOME INHIBITOR AND USES THEREOF 药捷安康(南京)科技股份有限公司 2023-07-13 WO disclosed