SCHEMBL2583067

SCHEMBL2583067

CN(CC(=O)N[C@@H](Cc1ccc(O)cc1)C(N)=O)C(=O)OC(C)(C)C

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CTSS P25774 1/20 0.46
CTSK P43235 1/20 0.46
ACE P12821 4/20 0.45
PTPN2 P17706 1/20 0.44
PTPN1 P18031 1/20 0.44
REN P00797 1/20 0.43
HPGDS O60760 3/20 0.43
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42
CA9 Q16790 1/20 0.42
MDM4 O15151 1/20 0.42
MDM2 Q00987 1/20 0.42
LY96 Q9Y6Y9 1/20 0.40
PRSS1 P07477 1/20 0.40
TPSAB1 Q15661 1/20 0.40
LNPEP Q9UIQ6 1/20 0.39
LHCGR P22888 1/20 0.39
NPY1R P25929 1/20 0.39
NPY2R P49146 1/20 0.39
NPY4R P50391 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2583065 1.00 CTSS (0.46) CTSSCTSKACEPTPN2PTPN1
SCHEMBL2585648 0.89 MDM4 (0.55) CTSSCTSKMDM4MDM2LY96
SCHEMBL2585645 0.89 MDM4 (0.55) CTSSCTSKMDM4MDM2LY96
SCHEMBL9564886 0.86 REN (0.42) CTSSCTSKACERENHPGDS
SCHEMBL2803528 0.80 CTSS (0.66) CTSSCTSKACEREN
SCHEMBL2801456 0.80 CTSS (0.66) CTSSCTSKACEREN
SCHEMBL2583010 0.79 TACR1 (0.51) ACE
SCHEMBL2583014 0.79 TACR1 (0.51) ACE
SCHEMBL18569864 0.75 KLK5 (0.46) MDM4MDM2LNPEP
SCHEMBL18257097 0.75 ESRRG (0.52) CA1PRSS1TPSAB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8350077-B2 Amides of creatine, method of their preparation, and remedy possessing a neuroprotective activity VERTEX CLOSED JOINT STOCK COMPANY (RU) 2013-01-08 US disclosed
US-20110269986-A1 AMIDES OF CREATNE, METHOD OF THEIR PREPARATION, AND REMEDY POSSESSING A NEUROPROTECTIVE ACTIVITY AMIDE BEVERAGE COMPANY, LLC 2011-11-03 US disclosed