SCHEMBL2585694

SCHEMBL2585694

C1=NCCC(c2ccc3nc(OC4CCN(Cc5ccccc5)CC4)sc3c2)=C1

nearest known ligand 0.42

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 7/20 0.42
CHEK2 O96017 1/20 0.41
ROCK1 Q13464 2/20 0.41
ROCK2 O75116 1/20 0.41
CCR2 P41597 1/20 0.41
BCHE P06276 2/20 0.40
ACHE P22303 2/20 0.40
KCNH2 Q12809 5/20 0.39
DRD2 P14416 1/20 0.39
HRH3 Q9Y5N1 1/20 0.38
SMN1; SMN2 Q16637 2/20 0.37
GAA P10253 1/20 0.37
OPRK1 P41145 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2594050 0.82 CHEK2 (0.42) LTA4HCHEK2ROCK1ROCK2CCR2
SCHEMBL16005681 0.80 LTA4H (0.45) LTA4HCHEK2ROCK1ROCK2CCR2
SCHEMBL2592883 0.79 LTA4H (0.48) LTA4HCHEK2ROCK1ROCK2CCR2
SCHEMBL12178006 0.77 NAMPT (0.44) LTA4HCHEK2BCHEACHEKCNH2
SCHEMBL2585277 0.76 GPR119 (0.57) LTA4HCHEK2BCHEACHEDRD2
SCHEMBL14731949 0.74 BCHE (0.38) LTA4HCHEK2ROCK1ROCK2CCR2
SCHEMBL14728992 0.73 GPR119 (0.47) LTA4HCHEK2BCHEACHEKCNH2
SCHEMBL8088919 0.64 HRH3 (0.52) ROCK1ROCK2CCR2ACHEKCNH2
SCHEMBL4855546 0.63 HRH3 (0.74) ROCK1ROCK2CCR2ACHEDRD2
SCHEMBL14718387 0.62 QDPR (0.36) CHEK2SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2566860-A1 BICYCLIC HETEROARYL COMPOUNDS AS GPR119 MODULATORS Bristol-Myers Squibb Company (US) 2013-03-13 EP disclosed
WO-2011140160-A1 BICYCLIC HETEROARYL COMPOUNDS AS GPR119 MODULATORS BRISTOL-MYERS SQUIBB COMPANY (US) 2011-11-10 WO disclosed