SCHEMBL25857067

SCHEMBL25857067

C=Cc1ccc(-c2nnc(N)c3ccccc23)c(O)c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.43
ESR1 P03372 1/20 0.34
ESR2 Q92731 1/20 0.34
NR1I2 O75469 3/20 0.33
SMARCA2 P51531 3/20 0.33
SMARCA4 P51532 3/20 0.33
PBRM1 Q86U86 3/20 0.33
TRPA1 O75762 1/20 0.33
BRD4 O60885 1/20 0.33
KMT2A Q03164 2/20 0.32
MEN1 O00255 1/20 0.32
CCNB2 O95067 2/20 0.32
CDK1 P06493 2/20 0.32
CCNB1 P14635 2/20 0.32
GSK3A P49840 2/20 0.32
GSK3B P49841 2/20 0.32
CDK5 Q00535 2/20 0.32
CDK5R1 Q15078 2/20 0.32
CCNB3 Q8WWL7 2/20 0.32
KRAS P01116 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25857052 0.80 ALDH1A1 (0.46) ESR1ESR2TRPA1
SCHEMBL24855423 0.74 KDM4E (0.43) KDM4E
SCHEMBL27352762 0.74 KDM4E (0.43) KDM4EESR1ESR2NR1I2SMARCA2
SCHEMBL25854476 0.74 KDM4E (0.43) KDM4EESR1ESR2NR1I2SMARCA2
SCHEMBL25861170 0.74 KDM4E (0.40) KDM4EESR1ESR2
SCHEMBL25856433 0.72 KDM4E (0.41) KDM4EESR1ESR2NR1I2SMARCA2
SCHEMBL27355770 0.72 KDM4E (0.41) KDM4EESR1ESR2NR1I2SMARCA2
SCHEMBL25861298 0.72 KDM4E (0.41) KDM4EESR1ESR2NR1I2SMARCA2
SCHEMBL25861928 0.71 TRPA1 (0.36) KDM4EESR1ESR2TRPA1KMT2A
SCHEMBL29502822 0.70 TRPA1 (0.52) KDM4EESR1ESR2TRPA1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023131277-A1 NLRP3 INFLAMMASOME INHIBITOR AND USES THEREOF 药捷安康(南京)科技股份有限公司 2023-07-13 WO disclosed