SCHEMBL25857052

SCHEMBL25857052

C=Cc1ccc(-c2nnc(NC)c3ccccc23)c(O)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.46
MAPT P10636 4/20 0.37
GAA P10253 2/20 0.37
PDK1 Q15118 2/20 0.35
PDK2 Q15119 1/20 0.35
PDK3 Q15120 1/20 0.35
PDK4 Q16654 1/20 0.35
NPSR1 Q6W5P4 2/20 0.35
TRPA1 O75762 1/20 0.34
MPO P05164 2/20 0.34
ENPP3 O14638 3/20 0.33
KLK7 P49862 1/20 0.33
KLK14 Q9P0G3 1/20 0.33
LMNA P02545 2/20 0.33
NPC1 O15118 1/20 0.32
NFKB1 P19838 1/20 0.32
RAB9A P51151 1/20 0.32
NFKB2 Q00653 1/20 0.32
RELA Q04206 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25855668 0.82 NLRP3 (0.47) ALDH1A1MAPTGAALMNA
SCHEMBL25857067 0.80 KDM4E (0.43) TRPA1ESR1ESR2
SCHEMBL25864315 0.77 NLRP3 (0.39) ALDH1A1MAPTGAATRPA1MPO
SCHEMBL25856769 0.76 ALDH1A1 (0.46) ALDH1A1MAPTGAAPDK1PDK2
SCHEMBL25861294 0.76 ALDH1A1 (0.43) ALDH1A1MAPTGAAPDK1PDK2
SCHEMBL25300751 0.76 NLRP3 (0.62)
SCHEMBL25300752 0.76 NLRP3 (0.62)
SCHEMBL25858838 0.75 ALDH1A1 (0.45) ALDH1A1MAPTGAAPDK1PDK2
SCHEMBL25861920 0.72 NLRP3 (0.39) TRPA1APPESR1ESR2
SCHEMBL29502822 0.67 TRPA1 (0.52) ALDH1A1MAPTGAANPSR1TRPA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023131277-A1 NLRP3 INFLAMMASOME INHIBITOR AND USES THEREOF 药捷安康(南京)科技股份有限公司 2023-07-13 WO disclosed