SCHEMBL25859182

SCHEMBL25859182

CCOCOc1cc(C#CC2CC2)ccc1-c1nnc(N)cc1C

nearest known ligand 0.35

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 2/20 0.35
CHRNA2 Q15822 2/20 0.35
CHRNB4 P30926 1/20 0.35
CHRNA3 P32297 1/20 0.35
CHRNA4 P43681 1/20 0.35
BACE1 P56817 12/20 0.33
APP P05067 2/20 0.32
PDGFRB P09619 1/20 0.32
PDGFRA P16234 1/20 0.32
PIKFYVE Q9Y2I7 2/20 0.31
GPR84 Q9NQS5 2/20 0.31
CACNA2D1 P54289 1/20 0.31
REN P00797 1/20 0.30
CTSD P07339 1/20 0.30
CYP3A4 P08684 1/20 0.30
BACE2 Q9Y5Z0 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25859156 0.84 CHRNB2 (0.37) CHRNB2CHRNA2CHRNB4CHRNA3CHRNA4
SCHEMBL31496024 0.84 CACNA2D1 (0.31) CACNA2D1
SCHEMBL25863128 0.79 CHRNB2 (0.36) CHRNB2CHRNA2CHRNB4CHRNA3CHRNA4
SCHEMBL25859817 0.78
SCHEMBL25303044 0.77 IL1B (0.53)
SCHEMBL25303047 0.77 IL1B (0.53)
SCHEMBL25861833 0.77 MEN1 (0.31) CACNA2D1
SCHEMBL31314084 0.76 ALDH1A1 (0.39) CACNA2D1
SCHEMBL25859343 0.76 ALDH1A1 (0.39) CACNA2D1
SCHEMBL31314309 0.75

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023131277-A1 NLRP3 INFLAMMASOME INHIBITOR AND USES THEREOF 药捷安康(南京)科技股份有限公司 2023-07-13 WO disclosed