SCHEMBL25859156

SCHEMBL25859156

CCOCOc1cc(C#CC2CC2)ccc1-c1nnc(N)nc1C

nearest known ligand 0.37

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 2/20 0.37
CHRNA2 Q15822 2/20 0.37
CHRNB4 P30926 1/20 0.37
CHRNA3 P32297 1/20 0.37
CHRNA4 P43681 1/20 0.37
PIKFYVE Q9Y2I7 2/20 0.34
BACE1 P56817 9/20 0.33
CACNA2D1 P54289 2/20 0.32
TBK1 Q9UHD2 1/20 0.32
APP P05067 2/20 0.32
PDGFRB P09619 1/20 0.32
PDGFRA P16234 1/20 0.32
TSHR P16473 1/20 0.31
GPR84 Q9NQS5 1/20 0.31
AKT1 P31749 1/20 0.30
ROCK1 Q13464 1/20 0.30
RPS6KA1 Q15418 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25859018 0.87 CACNA2D1 (0.34) CACNA2D1TSHR
SCHEMBL25863128 0.86 CHRNB2 (0.36) CHRNB2CHRNA2CHRNB4CHRNA3CHRNA4
SCHEMBL25859182 0.84 CHRNB2 (0.35) CHRNB2CHRNA2CHRNB4CHRNA3CHRNA4
SCHEMBL31314251 0.84 CACNA2D1 (0.33) CACNA2D1TSHR
SCHEMBL25857680 0.84 S1PR1 (0.36) CACNA2D1TSHR
SCHEMBL25859022 0.80 EGLN1 (0.37) PIKFYVEBACE1TBK1APP
SCHEMBL25299200 0.77 NLRP3 (0.40)
SCHEMBL25299201 0.77 NLRP3 (0.40)
SCHEMBL31314375 0.77 ALOX5AP (0.43)
SCHEMBL31314385 0.77 DHFR (0.40) CACNA2D1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023131277-A1 NLRP3 INFLAMMASOME INHIBITOR AND USES THEREOF 药捷安康(南京)科技股份有限公司 2023-07-13 WO disclosed