SCHEMBL25866294

SCHEMBL25866294

O=C1OC2(COC2)c2cc(Br)ccc21

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 1/20 0.43
OPRD1 P41143 1/20 0.43
NPY5R Q15761 2/20 0.39
TDP2 O95551 1/20 0.39
S100A4 P26447 1/20 0.37
PTPRC P08575 1/20 0.37
AVPR1A P37288 1/20 0.37
METAP1 P53582 1/20 0.37
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA4 P22748 1/20 0.36
CA7 P43166 1/20 0.36
CA9 Q16790 1/20 0.36
L3MBTL1 Q9Y468 2/20 0.36
TDP1 Q9NUW8 1/20 0.36
SIGMAR1 Q99720 1/20 0.35
AKR1C1 Q04828 1/20 0.35
MAPT P10636 2/20 0.35
MALT1 Q9UDY8 1/20 0.35
KDM4E B2RXH2 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29922337 0.94 OPRM1 (0.41) OPRM1OPRD1NPY5RTDP2S100A4
SCHEMBL31394738 0.87 AVPR1A (0.47) OPRM1OPRD1NPY5RTDP2S100A4
SCHEMBL18373219 0.82 OPRM1 (0.42) OPRM1OPRD1NPY5RTDP2S100A4
SCHEMBL25867610 0.80 TDP2 (0.39) TDP2AVPR1ACA7L3MBTL1TDP1
SCHEMBL18373156 0.80 NPY5R (0.45) OPRM1OPRD1NPY5RTDP2AVPR1A
SCHEMBL17586456 0.80 OPRM1 (0.40) OPRM1OPRD1NPY5RTDP2S100A4
SCHEMBL17586455 0.77 OPRM1 (0.41) OPRM1OPRD1NPY5RTDP2AVPR1A
SCHEMBL17586460 0.77 AVPR1A (0.48) OPRM1OPRD1NPY5RAVPR1ASIGMAR1
SCHEMBL31758718 0.77 NPY5R (0.36) OPRM1OPRD1NPY5RTDP2PTPRC
SCHEMBL31178327 0.77 SIGMAR1 (0.54) NPY5RAVPR1ATDP1SIGMAR1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023134656-A1 PEPTIDYL NITRILE COMPOUND AND USE THEREOF 上海壹典医药科技开发有限公司 2023-07-20 WO disclosed