SCHEMBL25866514

SCHEMBL25866514

CCOC(=O)CCCNC1(C(=O)OC)CC1

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.43
EPHX2 P34913 10/20 0.40
TSHR P16473 1/20 0.39
MGAM O43451 1/20 0.38
GAA P10253 1/20 0.38
SI P14410 1/20 0.38
MGAM2 Q2M2H8 1/20 0.38
SMYD3 Q9H7B4 1/20 0.38
TOP2A P11388 1/20 0.37
CYP3A4 P08684 1/20 0.36
CYP2C19 P33261 1/20 0.36
NR1I2 O75469 1/20 0.36
PGR P06401 1/20 0.36
ADORA3 P0DMS8 1/20 0.36
PTGS2 P35354 1/20 0.36
PDE4D Q08499 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22980572 0.92 CYP1A2 (0.44) CYP1A2EPHX2TSHRMGAMGAA
SCHEMBL8643850 0.86 TSHR (0.44) CYP1A2EPHX2TSHRMGAMGAA
SCHEMBL23007925 0.86 CYP1A2 (0.42) CYP1A2EPHX2TSHRMGAMGAA
SCHEMBL31327398 0.86 CYP1A2 (0.44) CYP1A2EPHX2TSHRMGAMGAA
SCHEMBL8640267 0.85 TSHR (0.46) CYP1A2EPHX2TSHRMGAMGAA
SCHEMBL29186867 0.81 TSHR (0.45) EPHX2TSHR
SCHEMBL8878481 0.79 TSHR (0.46) CYP1A2EPHX2TSHRMGAMGAA
SCHEMBL8716878 0.76 GAA (0.36) CYP1A2EPHX2TSHRMGAMGAA
SCHEMBL28023901 0.76 NPSR1 (0.35)
SCHEMBL8640882 0.75 TSHR (0.39) CYP1A2EPHX2TSHRMGAMGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4466266-B1 FUSED HETEROCYCLES AS 5-HT2A RECEPTOR AGONISTS TRANSNEURAL THERAPEUTICS INC (US) 2026-04-08 EP disclosed
US-12486268-B2 Fused heterocycles as 5-HT2A receptor agonists Transneural Therapeutics, Inc. (US) 2025-12-02 US disclosed
US-12459944-B2 Fused heterocycles as 5-HT2A receptor agonists Transneural Therapeutics, Inc. (US) 2025-11-04 US disclosed
US-20250243199-A1 FUSED HETEROCYCLES AS 5-HT2A RECEPTOR AGONISTS Transneural Therapeutics, Inc. (US) 2025-07-31 US disclosed
US-20240425503-A1 FUSED HETEROCYCLES AS 5-HT2A RECEPTOR AGONISTS Transneural Therapeutics, Inc. 2024-12-26 US disclosed
EP-4466266-A1 FUSED HETEROCYCLES AS 5-HT2A RECEPTOR AGONISTS Transneural Therapeutics, Inc. (US) 2024-11-27 EP disclosed
WO-2023141225-A1 FUSED HETEROCYCLES AS 5-HT2A RECEPTOR AGONISTS ONSERO THERAPEUTICS INC. (US) 2023-07-27 WO disclosed
WO-2023141225-A1 FUSED HETEROCYCLES AS 5-HT2A RECEPTOR AGONISTS ONSERO THERAPEUTICS INC. (US) 2023-07-27 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12459944-B2 Fused heterocycles as 5-HT2A receptor agonists HTR2A, HTR2C, HTR5A CYP1A2 125/4885EPHX2 588/4885TSHR 248/4885
US-20250243199-A1 FUSED HETEROCYCLES AS 5-HT2A RECEPTOR AGONISTS HTR2A, HTR2C, HTR5A CYP1A2 125/4885EPHX2 588/4885TSHR 248/4885
US-20240425503-A1 FUSED HETEROCYCLES AS 5-HT2A RECEPTOR AGONISTS HTR2A, HTR2C, HTR1A CYP1A2 113/4885EPHX2 742/4885TSHR 227/4885
US-12486268-B2 Fused heterocycles as 5-HT2A receptor agonists HTR2A, HTR2C, HTR5A CYP1A2 125/4885EPHX2 588/4885TSHR 248/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.