SCHEMBL25880000

SCHEMBL25880000

CN1CCN(CCNC(=O)c2cc(Nc3ncc4ccccc4n3)c[nH]2)CC1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRAF P15056 2/20 0.46
USP2 O75604 1/20 0.44
MAP3K5 Q99683 1/20 0.43
HTR1A P08908 4/20 0.42
POLR1A O95602 1/20 0.42
KDM4E B2RXH2 2/20 0.42
HSD17B10 Q99714 2/20 0.42
SMN1; SMN2 Q16637 1/20 0.41
KDM5B Q9UGL1 1/20 0.41
ALDH1A1 P00352 1/20 0.41
MAP4K1 Q92918 1/20 0.40
DRD2 P14416 1/20 0.40
PDGFRB P09619 1/20 0.40
PDGFRA P16234 1/20 0.40
RAD52 P43351 1/20 0.40
CYP1A2 P05177 1/20 0.40
MAPT P10636 1/20 0.40
CYP2C9 P11712 1/20 0.40
EGFR P00533 1/20 0.40
AXL P30530 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30512121 1.00 BRAF (0.46) BRAFUSP2MAP3K5HTR1APOLR1A
SCHEMBL25880004 0.85 SYK (0.45) MAP3K5MAP4K1
SCHEMBL30512114 0.83 EGFR (0.48) MAP3K5MAP4K1EGFRAXL
SCHEMBL25882002 0.83 EGFR (0.48) MAP3K5MAP4K1EGFRAXL
SCHEMBL25879895 0.83 BRAF (0.51) BRAFMAP3K5RAD52
SCHEMBL30512108 0.83 BRAF (0.51) BRAFMAP3K5RAD52
SCHEMBL25879889 0.83 HRH4 (0.50) MAP3K5MAP4K1PDGFRBPDGFRA
SCHEMBL30512112 0.79 MAP3K5 (0.54) BRAFMAP3K5
SCHEMBL25879550 0.79 MAP3K5 (0.54) BRAFMAP3K5
SCHEMBL30512136 0.76 MAP3K5 (0.54) BRAFMAP3K5SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023138412-A1 FUSED PYRIMIDIN-2-AMINE COMPOUNDS AS CDK20 INHIBITORS INSILICO MEDICINE IP LIMITED (CN) 2023-07-27 WO disclosed