SCHEMBL25882002

SCHEMBL25882002

CN1CCC(NC(=O)c2cc(Nc3ncc4ccccc4n3)c[nH]2)CC1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 1/20 0.48
MAPK1 P28482 1/20 0.47
AURKA O14965 3/20 0.45
AURKB Q96GD4 2/20 0.45
MAP3K5 Q99683 1/20 0.44
IGF1R P08069 2/20 0.44
MAP4K1 Q92918 2/20 0.44
SELP P16109 1/20 0.43
TYRO3 Q06418 1/20 0.43
CCNA2 P20248 2/20 0.43
CDK2 P24941 2/20 0.43
CCNA1 P78396 2/20 0.43
WEE1 P30291 1/20 0.43
PLK1 P53350 1/20 0.43
SYK P43405 1/20 0.43
BRD4 O60885 3/20 0.43
JAK2 O60674 1/20 0.43
NTRK1 P04629 1/20 0.43
NTRK3 Q16288 1/20 0.43
NTRK2 Q16620 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30512114 1.00 EGFR (0.48) EGFRMAPK1AURKAAURKBMAP3K5
SCHEMBL25880004 0.86 SYK (0.45) MAP3K5IGF1RMAP4K1TYRO3SYK
SCHEMBL30512121 0.83 BRAF (0.46) EGFRMAP3K5MAP4K1AXL
SCHEMBL25880000 0.83 BRAF (0.46) EGFRMAP3K5MAP4K1AXL
SCHEMBL25879889 0.82 HRH4 (0.50) MAP3K5MAP4K1CDK2WEE1SYK
SCHEMBL30512112 0.81 MAP3K5 (0.54) MAPK1AURKAMAP3K5CDK2SYK
SCHEMBL25879550 0.81 MAP3K5 (0.54) MAPK1AURKAMAP3K5CDK2SYK
SCHEMBL25880449 0.78 HRH4 (0.53) MAP3K5CCNA2CDK2AXL
SCHEMBL25880130 0.77 MAP4K1 (0.45) MAP3K5MAP4K1
SCHEMBL30512136 0.77 MAP3K5 (0.54) MAPK1AURKAMAP3K5CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023138412-A1 FUSED PYRIMIDIN-2-AMINE COMPOUNDS AS CDK20 INHIBITORS INSILICO MEDICINE IP LIMITED (CN) 2023-07-27 WO disclosed