SCHEMBL25894839

SCHEMBL25894839

CNc1ccc(C(F)(F)C(F)(F)F)nc1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 1/20 0.37
TRPV4 Q9HBA0 1/20 0.35
CYP2C9 P11712 1/20 0.35
SLC22A6 Q4U2R8 1/20 0.35
SLC22A8 Q8TCC7 1/20 0.35
SLC22A12 Q96S37 1/20 0.35
SLC22A11 Q9NSA0 1/20 0.35
CA12 O43570 3/20 0.34
CA1 P00915 3/20 0.34
CA2 P00918 3/20 0.34
RRM2 P31350 1/20 0.33
ABCC9 O60706 1/20 0.33
ABCC8 Q09428 1/20 0.33
KCNJ11 Q14654 1/20 0.33
KCNJ8 Q15842 1/20 0.33
ABL1 P00519 1/20 0.33
BCR P11274 1/20 0.33
EGFR P00533 2/20 0.33
EPHX2 P34913 1/20 0.32
CA4 P22748 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8171100 0.84 TRPV4 (0.52) KIF11TRPV4CYP2C9SLC22A6SLC22A8
SCHEMBL23055282 0.82 SLC22A12 (0.39) KIF11TRPV4CYP2C9SLC22A6SLC22A8
Hydrochloric Acid SCHEMBL29162081 0.82 TRPV4 (0.50) KIF11TRPV4CYP2C9SLC22A6SLC22A8
Hydrochloric Acid SCHEMBL29162116 0.81 SLC22A12 (0.38) KIF11TRPV4CYP2C9SLC22A6SLC22A8
SCHEMBL14283237 0.78 CA12 (0.38) KIF11TRPV4CYP2C9SLC22A6SLC22A8
SCHEMBL21016949 0.74 TGFBR1 (0.40) KIF11CYP2C9SLC22A6SLC22A8SLC22A12
SCHEMBL22601556 0.74 CA12 (0.35) KIF11TRPV4CYP2C9SLC22A6SLC22A8
SCHEMBL25894850 0.74 CCR1 (0.44) TRPV4PTGS2ALDH1A1
SCHEMBL30074800 0.72 TRPV4 (0.47) TRPV4CYP2C9SLC22A6SLC22A8SLC22A12
SCHEMBL22001498 0.70 CHRNA7 (0.43) CYP2C9CA12CA1CA2RRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20260103464-A1 CYCLOPROPYL-(HETERO)ARYL-SUBSTITUTED ETHYLSULPHONYL-PYRIDINE DERIVATIVES BOEHRINGER INGELHEIM VETMEDICA GMBH (DE) 2026-04-16 US disclosed
US-12435083-B2 Cyclopropyl-(hetero)aryl-substituted ethylsulphonyl-pyridine derivatives BOEHRINGER INGELHEIM VETMEDICA GMBH (DE) 2025-10-07 US disclosed
CN-118355004-A Cyclopropyl- (heteroaryl) -substituted ethylsulfonyl-pyridine derivatives 勃林格殷格翰动物保健有限公司 2024-07-16 CN disclosed
US-20230234951-A1 CYCLOPROPYL-(HETERO)ARYL-SUBSTITUTED ETHYLSULPHONYL-PYRIDINE DERIVATIVES BOEHRINGER INGELHEIM PHARMA GMBH & CO. KG (DE) 2023-07-27 US disclosed
US-20230234951-A1 CYCLOPROPYL-(HETERO)ARYL-SUBSTITUTED ETHYLSULPHONYL-PYRIDINE DERIVATIVES BOEHRINGER INGELHEIM PHARMA GMBH & CO. KG (DE) 2023-07-27 US disclosed
WO-2023036934-A1 CYCLOPROPYL-(HETERO)ARYL-SUBSTITUTED ETHYLSULPHONYLPYRIDINE DERIVATIVES BOEHRINGER INGELHEIM VETMEDICA GMBH (DE) 2023-03-16 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230234951-A1 CYCLOPROPYL-(HETERO)ARYL-SUBSTITUTED ETHYLSULPHONYL-PYRIDINE DERIVATIVES CYCS, CYP2E1, AHR KIF11 4545/4885TRPV4 2332/4885CYP2C9 24/4885
US-12435083-B2 Cyclopropyl-(hetero)aryl-substituted ethylsulphonyl-pyridine derivatives CYCS, CYP2E1, CYP1A1 KIF11 4564/4885TRPV4 2151/4885CYP2C9 21/4885
US-20260103464-A1 CYCLOPROPYL-(HETERO)ARYL-SUBSTITUTED ETHYLSULPHONYL-PYRIDINE DERIVATIVES CBR3, CYCS, CBR1 KIF11 4231/4885TRPV4 2718/4885CYP2C9 433/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.