SCHEMBL25899947

SCHEMBL25899947

CCc1ccc2c(n1)N(CC)C(=O)C2(C)C

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MARK3 P27448 1/20 0.50
PDE4B Q07343 2/20 0.41
PDE4A P27815 1/20 0.41
PDE4C Q08493 1/20 0.41
PDE4D Q08499 1/20 0.41
AURKA O14965 2/20 0.34
AURKB Q96GD4 2/20 0.34
ELANE P08246 1/20 0.33
PGR P06401 1/20 0.32
BACE1 P56817 1/20 0.31
BACE2 Q9Y5Z0 1/20 0.31
CHEK1 O14757 1/20 0.31
SRC P12931 1/20 0.31
CDK2 P24941 1/20 0.31
KDR P35968 1/20 0.31
FLT3 P36888 1/20 0.31
GSK3B P49841 1/20 0.31
PDE3A Q14432 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
BRD4 O60885 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25898322 0.81 MARK3 (0.50) MARK3AURKAAURKBELANEPGR
SCHEMBL25888905 0.79 MARK3 (0.48) MARK3AURKAAURKBELANEPGR
SCHEMBL25899645 0.79 MARK3 (0.48) MARK3AURKAAURKBELANEPGR
SCHEMBL18719875 0.67 AURKA (0.40) MARK3AURKAAURKBELANEPGR
SCHEMBL23097108 0.66 PDK2 (0.47) MARK3PDE4BPDE4APDE4CPDE4D
SCHEMBL9202873 0.65 GPR55 (0.56) MARK3ELANE
SCHEMBL10953690 0.64 ELANE (0.50) MARK3AURKAAURKBELANEBACE1
SCHEMBL17275707 0.64 ALDH1A1 (0.47) MARK3AURKAAURKBPGRBACE1
SCHEMBL4501318 0.64 ATAD2 (0.44) MARK3AURKAAURKBELANEPGR
SCHEMBL5543415 0.61 CYP2C9 (0.49) AURKAAURKBCHEK1SRCCDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023138362-A1 WEE1 INHIBITOR, PREPARATION THEREFOR, AND USE THEREOF 江苏天士力帝益药业有限公司 2023-07-27 WO disclosed