SCHEMBL25898322

SCHEMBL25898322

CCN1C(=O)C(C)(C)c2ccc(Br)nc21

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
MARK3 P27448 1/20 0.50
AURKA O14965 1/20 0.34
AURKB Q96GD4 1/20 0.34
ELANE P08246 1/20 0.33
CNR1 P21554 1/20 0.33
PGR P06401 2/20 0.32
BACE1 P56817 1/20 0.31
BACE2 Q9Y5Z0 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
ALDH1A1 P00352 1/20 0.30
PKM P14618 1/20 0.30
KMT2A Q03164 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
MAPT P10636 1/20 0.30
BRD4 O60885 1/20 0.30
CYP1B1 Q16678 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25888905 0.82 MARK3 (0.48) MARK3AURKAAURKBELANEPGR
SCHEMBL25899947 0.81 MARK3 (0.50) MARK3AURKAAURKBELANEPGR
SCHEMBL25899645 0.79 MARK3 (0.48) MARK3AURKAAURKBELANEPGR
SCHEMBL17275707 0.70 ALDH1A1 (0.47) MARK3AURKAAURKBCNR1PGR
SCHEMBL25898318 0.70 USP1 (0.38) ALDH1A1KMT2AMAPTBRD4
SCHEMBL32681245 0.68 SMN1; SMN2 (0.34) KMT2ASMN1; SMN2
SCHEMBL9202873 0.65 GPR55 (0.56) MARK3ELANECNR1ALDH1A1KMT2A
SCHEMBL10953690 0.64 ELANE (0.50) MARK3AURKAAURKBELANECNR1
SCHEMBL4501318 0.64 ATAD2 (0.44) MARK3AURKAAURKBELANECNR1
SCHEMBL18719875 0.64 AURKA (0.40) MARK3AURKAAURKBELANECNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023138362-A1 WEE1 INHIBITOR, PREPARATION THEREFOR, AND USE THEREOF 江苏天士力帝益药业有限公司 2023-07-27 WO disclosed