SCHEMBL2594714

SCHEMBL2594714

O=C(O)Cc1nc(S(=O)(=O)Cc2ccccc2)c2ccccn12

nearest known ligand 0.64

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HCRTR2 O43614 5/20 0.64
PTGDR2 Q9Y5Y4 1/20 0.45
HCRTR1 O43613 4/20 0.43
ALDH1A1 P00352 5/20 0.42
MAPT P10636 4/20 0.42
KDM4E B2RXH2 2/20 0.42
MEN1 O00255 2/20 0.42
KMT2A Q03164 2/20 0.42
TSHR P16473 3/20 0.38
HSD17B10 Q99714 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
AKR1B1 P15121 1/20 0.37
GSR P00390 1/20 0.36
TXNRD1 Q16881 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
MMP1 P03956 1/20 0.36
MMP2 P08253 1/20 0.36
MMP9 P14780 1/20 0.36
MMP8 P22894 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7706361 0.85 HCRTR2 (0.62) HCRTR2HCRTR1ALDH1A1MAPTKDM4E
SCHEMBL7709292 0.79 HCRTR2 (1.00) HCRTR2HCRTR1ALDH1A1MAPTKMT2A
SCHEMBL7708524 0.78 HCRTR2 (0.74) HCRTR2HCRTR1LMNAPOLB
SCHEMBL2594821 0.76 HCRTR2 (0.50) HCRTR2HCRTR1ALDH1A1MAPTKDM4E
SCHEMBL12480878 0.71 KMT2A (0.47) HCRTR2PTGDR2ALDH1A1MAPTKDM4E
SCHEMBL2585096 0.71 HCRTR2 (0.74) HCRTR2PTGDR2HCRTR1ALDH1A1MAPT
SCHEMBL15485100 0.70 KMT2A (0.43) HCRTR2PTGDR2ALDH1A1MAPTKDM4E
SCHEMBL31214657 0.68 KDM4E (0.55) PTGDR2ALDH1A1MAPTKDM4EMEN1
SCHEMBL7708626 0.66 HCRTR1 (0.71) HCRTR2PTGDR2HCRTR1ALDH1A1MAPT
SCHEMBL31282458 0.64 ALDH1A1 (0.45) PTGDR2ALDH1A1MAPTKDM4EMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011138266-A1 INDOLIZINE AND IMIDAZOPYRIDINE DERIVATIVES AS OREXIN RECEPTOR ANTAGONISTS EVOTEC AG (DE) 2011-11-10 WO disclosed
WO-2011138266-A1 INDOLIZINE AND IMIDAZOPYRIDINE DERIVATIVES AS OREXIN RECEPTOR ANTAGONISTS EVOTEC AG (DE) 2011-11-10 WO disclosed