SCHEMBL7708524

SCHEMBL7708524

CN(Cc1cccc(Cl)c1)C(=O)Cc1nc(S(=O)(=O)Cc2ccccc2)c2ccccn12

nearest known ligand 0.74

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HCRTR2 O43614 6/20 0.74
HCRTR1 O43613 5/20 0.52
AOC3 Q16853 3/20 0.42
LMNA P02545 1/20 0.42
POLB P06746 1/20 0.40
TSPO P30536 1/20 0.39
RIPK1 Q13546 1/20 0.39
TP53 P04637 1/20 0.38
GABRA1 P14867 1/20 0.38
GABRA5 P31644 1/20 0.38
GABRB2 P47870 1/20 0.38
PIN1 Q13526 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7709292 0.85 HCRTR2 (1.00) HCRTR2HCRTR1LMNATSPOTP53
SCHEMBL7707649 0.80 HCRTR2 (0.82) HCRTR2HCRTR1AOC3LMNAPOLB
SCHEMBL2594714 0.78 HCRTR2 (0.64) HCRTR2HCRTR1LMNAPOLB
SCHEMBL7707208 0.76 HCRTR2 (0.81) HCRTR2HCRTR1AOC3LMNAPOLB
SCHEMBL7706361 0.76 HCRTR2 (0.62) HCRTR2HCRTR1LMNA
SCHEMBL7709056 0.75 HCRTR2 (0.82) HCRTR2HCRTR1AOC3LMNATSPO
SCHEMBL7707551 0.73 HCRTR2 (0.71) HCRTR2HCRTR1AOC3LMNATSPO
SCHEMBL7702437 0.71 HCRTR1 (0.81) HCRTR2HCRTR1LMNAPOLBTP53
SCHEMBL7712431 0.71 HCRTR2 (0.66) HCRTR2HCRTR1AOC3LMNAPOLB
SCHEMBL7707423 0.69 HCRTR2 (1.00) HCRTR2HCRTR1POLBTSPO

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011138266-A1 INDOLIZINE AND IMIDAZOPYRIDINE DERIVATIVES AS OREXIN RECEPTOR ANTAGONISTS EVOTEC AG (DE) 2011-11-10 WO disclosed