SCHEMBL25947313

SCHEMBL25947313

CCOC(=O)c1c(CNC(=O)OC(C)(C)C)n(C)c2cc(-c3cccc4ccccc34)c(C3CCCC3)cc12

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 2/20 0.38
KDM4E B2RXH2 3/20 0.37
PKM P14618 1/20 0.36
RAD52 P43351 1/20 0.36
TSHR P16473 1/20 0.35
ALOX5 P09917 2/20 0.35
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
MAPT P10636 2/20 0.35
P4HB P07237 1/20 0.35
ALDH1A1 P00352 1/20 0.34
SPR P35270 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
CNR2 P34972 1/20 0.34
CACNA1C Q13936 1/20 0.34
KDM4A O75164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25947740 0.97 PKM (0.38) CASP3KDM4EPKMRAD52TSHR
SCHEMBL25947210 0.97 KDM4E (0.38) CASP3KDM4EPKMRAD52TSHR
SCHEMBL25939754 0.88 CASP3 (0.39) CASP3KDM4EPKMRAD52TSHR
SCHEMBL25947076 0.88 TSHR (0.38) CASP3KDM4ERAD52TSHRALOX5
SCHEMBL25947609 0.87 TSHR (0.36) CASP3KDM4ERAD52TSHRALOX5
SCHEMBL25946423 0.86 ALOX5 (0.42) KDM4ERAD52ALOX5MEN1KMT2A
SCHEMBL25946906 0.86 RAD52 (0.44) KDM4EPKMRAD52TSHRALOX5
SCHEMBL25948949 0.85 CASP3 (0.39) CASP3KDM4EPKMRAD52TSHR
SCHEMBL25939765 0.85 KDM4E (0.39) CASP3KDM4EPKMRAD52TSHR
SCHEMBL25947315 0.85 TSHR (0.41) CASP3KDM4EPKMTSHRALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4209492-A1 COMPOUND FOR TREATING THROMBOTIC DISEASES Shanghai Institute of Materia Medica, Chinese Academy of Sciences (CN) 2023-07-12 EP disclosed