SCHEMBL2595265

SCHEMBL2595265

Cc1noc(C2CCCCC2C(=O)NN)n1

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 1/20 0.40
FABP4 P15090 3/20 0.36
FABP5 Q01469 3/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
EPHX2 P34913 1/20 0.35
ALDH1A1 P00352 1/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
CCR5 P51681 1/20 0.35
CPT2 P23786 1/20 0.34
CPT1A P50416 1/20 0.34
HSD11B1 P28845 1/20 0.33
SCN9A Q15858 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2593261 0.82 CPT2 (0.48) CHRM2FABP4FABP5SMN1; SMN2EPHX2
SCHEMBL2595298 0.78 SMN1; SMN2 (0.36) FABP4FABP5SMN1; SMN2ALDH1A1CYP1A2
SCHEMBL2595542 0.76 ALDH1A1 (0.36) SMN1; SMN2ALDH1A1CYP1A2CYP3A4CYP2C9
SCHEMBL2595492 0.75 SMN1; SMN2 (0.36) FABP4FABP5SMN1; SMN2ALDH1A1CYP1A2
SCHEMBL2585944 0.74 CCR5 (0.43) CHRM2EPHX2CCR5HSD11B1
SCHEMBL2585948 0.74 CCR5 (0.43) CHRM2EPHX2CCR5HSD11B1
SCHEMBL2596228 0.73 SMN1; SMN2 (0.35) SMN1; SMN2ALDH1A1CYP1A2CYP3A4CYP2C9
SCHEMBL2596210 0.73 SMN1; SMN2 (0.35) SMN1; SMN2ALDH1A1CYP1A2CYP3A4CYP2C9
SCHEMBL2589850 0.72 ALDH1A1 (0.38) SMN1; SMN2ALDH1A1CYP1A2CYP3A4CYP2C9
SCHEMBL2596225 0.72 HCRTR1 (0.35) FABP4FABP5SMN1; SMN2ALDH1A1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2569319-A1 HETEROARYL-CYCLOHEXYL-TETRAAZABENZO[E]AZULENES F.HOFFMANN-LA ROCHE AG (CH) 2013-03-20 EP disclosed
WO-2011141396-A1 HETEROARYL-CYCLOHEXYL-TETRAAZABENZO[E]AZULENES F. HOFFMANN-LA ROCHE AG (CH) 2011-11-17 WO disclosed