SCHEMBL2595618

SCHEMBL2595618

O=S(=O)(NCOc1ccccc1)c1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.55
MEN1 O00255 2/20 0.54
KMT2A Q03164 2/20 0.54
HTT P42858 1/20 0.54
KEAP1 Q14145 1/20 0.53
KDM4E B2RXH2 1/20 0.53
LMNA P02545 1/20 0.53
PKM P14618 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
TBXA2R P21731 1/20 0.50
TBXAS1 P24557 1/20 0.50
GAA P10253 1/20 0.50
MAPT P10636 2/20 0.49
AR P10275 1/20 0.49
MAPK1 P28482 1/20 0.49
GBA1 P04062 1/20 0.49
POLB P06746 1/20 0.48
PGR P06401 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7572313 0.88 CA12 (0.59) ALDH1A1MEN1KMT2AHTTSMN1; SMN2
SCHEMBL7571617 0.88 TAAR1 (0.56) ALDH1A1MEN1KMT2AHTTPKM
SCHEMBL7573869 0.87 MEN1 (0.54) ALDH1A1MEN1KMT2AHTTTBXA2R
SCHEMBL7570427 0.84 AR (0.57) ALDH1A1MEN1KMT2AHTTLMNA
SCHEMBL7570456 0.84 MEN1 (0.51) ALDH1A1MEN1KMT2AHTTKDM4E
SCHEMBL411104 0.81 ALDH1A1 (0.79) ALDH1A1MEN1KMT2AHTTKDM4E
SCHEMBL7580123 0.81 PGR (0.57) ALDH1A1MEN1KMT2AHTTLMNA
SCHEMBL1880968 0.80 ALDH1A1 (0.72) ALDH1A1MEN1KMT2AHTTKDM4E
SCHEMBL1876555 0.79 ALDH1A1 (0.71) ALDH1A1MEN1KMT2AHTTKDM4E
SCHEMBL19280574 0.78 ALDH1A1 (0.56) ALDH1A1KEAP1KDM4ELMNAPKM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2563770-A1 BIARYL PHOSPHODIESTERASE INHIBITORS Leo Pharma A/S (DK) 2013-03-06 EP disclosed
WO-2011134468-A1 BIARYL PHOSPHODIESTERASE INHIBITORS LEO PHARMA A/S (DK) 2011-11-03 WO disclosed