SCHEMBL25959229

SCHEMBL25959229

N=C(Br)c1cnc(C(=O)N2CCC(O)CC2)cc1NCC(F)(F)F

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PCSK9 Q8NBP7 1/20 0.39
SCN9A Q15858 4/20 0.38
CNR2 P34972 2/20 0.35
VNN1 O95497 1/20 0.35
ALOX5AP P20292 2/20 0.35
FEN1 P39748 2/20 0.35
LRRK2 Q5S007 3/20 0.34
TRPC6 Q9Y210 2/20 0.33
IRAK4 Q9NWZ3 1/20 0.33
GPR52 Q9Y2T5 1/20 0.33
LIPE Q05469 1/20 0.33
MERTK Q12866 1/20 0.33
RORC P51449 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25959315 0.96 SCN9A (0.41) PCSK9SCN9ACNR2VNN1ALOX5AP
SCHEMBL25958904 0.88 ALDH1A1 (0.37) SCN9ACNR2VNN1LRRK2
SCHEMBL25959270 0.84 SCN9A (0.40) SCN9ACNR2VNN1LRRK2IRAK4
SCHEMBL25959288 0.84 VNN1 (0.41) SCN9ACNR2VNN1LRRK2RORC
SCHEMBL25958987 0.83 LRRK2 (0.41) SCN9AVNN1LRRK2RORC
SCHEMBL25960484 0.80 KMT2A (0.36) IRAK4
SCHEMBL25957156 0.80 ALDH1A1 (0.41)
SCHEMBL25958758 0.78 ALOX5AP (0.38) PCSK9ALOX5APFEN1TRPC6
SCHEMBL25960670 0.77 IRAK4 (0.36) IRAK4
SCHEMBL25960881 0.75 PCSK9 (0.34) PCSK9CNR2LRRK2TRPC6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3870582-B1 5-AZAINDAZOLE DERIVATIVES AS ADENOSINE RECEPTOR ANTAGONISTS MERCK PATENT GMBH (DE) 2023-07-19 EP disclosed