SCHEMBL25959288

SCHEMBL25959288

N=C(Br)c1cnc(C(=O)N2CCOCC(O)C2)cc1NCC(F)(F)F

nearest known ligand 0.41

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
VNN1 O95497 1/20 0.41
LRRK2 Q5S007 9/20 0.37
SMN1; SMN2 Q16637 1/20 0.32
CNR2 P34972 2/20 0.31
FLT3 P36888 1/20 0.31
RORC P51449 1/20 0.31
SCN9A Q15858 4/20 0.31
HPGD P15428 1/20 0.31
TSHR P16473 1/20 0.31
ESR2 Q92731 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25958987 0.85 LRRK2 (0.41) VNN1LRRK2SMN1; SMN2FLT3RORC
SCHEMBL25959229 0.84 PCSK9 (0.39) VNN1LRRK2CNR2RORCSCN9A
SCHEMBL25961687 0.82 VNN1 (0.39) VNN1LRRK2HPGD
SCHEMBL25959308 0.82 LRRK2 (0.36) VNN1LRRK2SMN1; SMN2CNR2RORC
SCHEMBL25957627 0.82 VNN1 (0.35) VNN1LRRK2
SCHEMBL25957185 0.82 VNN1 (0.38) VNN1SMN1; SMN2TSHR
SCHEMBL25957181 0.81 VNN1 (0.36) VNN1LRRK2
SCHEMBL25958792 0.81 VNN1 (0.40) VNN1SMN1; SMN2HPGDTSHRESR2
SCHEMBL25959315 0.80 SCN9A (0.41) VNN1LRRK2CNR2SCN9A
SCHEMBL25958904 0.80 ALDH1A1 (0.37) VNN1LRRK2CNR2SCN9AHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3870582-B1 5-AZAINDAZOLE DERIVATIVES AS ADENOSINE RECEPTOR ANTAGONISTS MERCK PATENT GMBH (DE) 2023-07-19 EP disclosed