SCHEMBL25958792

SCHEMBL25958792

N=C(Br)c1cnc(C(=O)N2CCOCC(O)C2)cc1N

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
VNN1 O95497 2/20 0.40
SMN1; SMN2 Q16637 1/20 0.37
HPGD P15428 1/20 0.34
TSHR P16473 1/20 0.34
ESR2 Q92731 1/20 0.34
GRM5 P41594 1/20 0.32
PDE4B Q07343 1/20 0.32
LMNA P02545 1/20 0.31
NPC1 O15118 1/20 0.31
RAB9A P51151 1/20 0.31
BTK Q06187 1/20 0.31
NTRK1 P04629 1/20 0.31
DPP4 P27487 1/20 0.30
KMT2A Q03164 1/20 0.30
BMPR1B O00238 1/20 0.30
BMPR1A P36894 1/20 0.30
TGFBR1 P36897 1/20 0.30
ACVRL1 P37023 1/20 0.30
ACVR1 Q04771 1/20 0.30
PIK3C3 Q8NEB9 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25958662 0.82 SMN1; SMN2 (0.45) VNN1SMN1; SMN2HPGDTSHRESR2
SCHEMBL25958553 0.82 VNN1 (0.43) VNN1SMN1; SMN2HPGDTSHRESR2
SCHEMBL25958758 0.81 ALOX5AP (0.38) ALOX5APFEN1
SCHEMBL25959288 0.81 VNN1 (0.41) VNN1SMN1; SMN2HPGDTSHRESR2
SCHEMBL25958820 0.77 SMN1; SMN2 (0.36) SMN1; SMN2HPGDTSHRESR2GRM5
SCHEMBL25958835 0.77 SCN9A (0.38) DPP4ALOX5APFEN1
SCHEMBL25958653 0.77 ALDH1A1 (0.42) HPGDTSHRNPC1RAB9ADPP4
SCHEMBL25958773 0.72 SCN9A (0.36) VNN1HPGDKMT2A
SCHEMBL24058957 0.72 ROCK2 (0.46) VNN1SMN1; SMN2HPGDTSHRESR2
SCHEMBL24058963 0.72 VNN1 (0.41) VNN1SMN1; SMN2HPGDTSHRESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3870582-B1 5-AZAINDAZOLE DERIVATIVES AS ADENOSINE RECEPTOR ANTAGONISTS MERCK PATENT GMBH (DE) 2023-07-19 EP disclosed