SCHEMBL25959425

SCHEMBL25959425

CC(F)(F)CNc1cc(C#N)ncc1C(N)Br

nearest known ligand 0.34

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CHEK1 O14757 4/20 0.34
IRAK4 Q9NWZ3 1/20 0.33
LRRK2 Q5S007 1/20 0.32
AR P10275 1/20 0.31
TBK1 Q9UHD2 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25959437 0.75 IRAK4 (0.39) CHEK1IRAK4AR
SCHEMBL24056640 0.59 CHEK1 (0.49) CHEK1
SCHEMBL25555781 0.57 GABRA1 (0.37) CHEK1
SCHEMBL22448681 0.57 LMNA (0.38) CHEK1
SCHEMBL31633801 0.57 GPR6 (0.37) CHEK1IRAK4LRRK2
SCHEMBL18266146 0.56 PDE2A (0.39)
SCHEMBL30773928 0.56 MBOAT4 (0.37) IRAK4AR
SCHEMBL22023351 0.56 MBOAT4 (0.37) IRAK4AR
SCHEMBL25144387 0.56 GABRP (0.36) CHEK1LRRK2AR
SCHEMBL3107926 0.56 UHRF1 (0.54) CHEK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3870582-B1 5-AZAINDAZOLE DERIVATIVES AS ADENOSINE RECEPTOR ANTAGONISTS MERCK PATENT GMBH (DE) 2023-07-19 EP disclosed