SCHEMBL25965347

SCHEMBL25965347

CC(=O)N1CC[C@@H](N(C)c2cccc(Br)c2)C1

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
OPRD1 P41143 1/20 0.43
L3MBTL3 Q96JM7 7/20 0.41
L3MBTL1 Q9Y468 4/20 0.41
L3MBTL4 Q8NA19 1/20 0.41
MBTD1 Q05BQ5 2/20 0.41
ALDH1A1 P00352 2/20 0.38
TP53 P04637 1/20 0.38
NPY5R Q15761 2/20 0.37
KMT5A Q9NQR1 1/20 0.37
CCR5 P51681 1/20 0.37
BRD4 O60885 1/20 0.37
CREBBP Q92793 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL25967729 0.92 OPRD1 (0.45) OPRD1L3MBTL3L3MBTL1L3MBTL4MBTD1
SCHEMBL25965344 0.83 USP30 (0.53)
SCHEMBL25965350 0.79 LIPG (0.36) L3MBTL3ALDH1A1NPY5RCCR5
SCHEMBL25967727 0.78 MEN1 (0.51)
SCHEMBL16391135 0.76 CASP6 (0.44) L3MBTL3NPY5R
SCHEMBL16698134 0.76 CASP6 (0.44) L3MBTL3NPY5R
SCHEMBL16698136 0.76 CASP6 (0.44) L3MBTL3NPY5R
SCHEMBL1419786 0.75 ALDH1A1 (0.39) L3MBTL3MBTD1ALDH1A1
SCHEMBL25356633 0.75 KDM1A (0.48) L3MBTL3L3MBTL1ALDH1A1NPY5R
SCHEMBL14242799 0.74 ALDH1A1 (0.38) L3MBTL3MBTD1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230357242-A1 COMPOUND AS AKT KINASE INHIBITOR CHIA TAI TIANQING PHARMACEUTICAL GROUP CO., LTD. (CN) 2023-11-09 US disclosed
EP-4223754-A1 COMPOUND AS AKT KINASE INHIBITOR CHIA TAI TIANQING PHARMACEUTICAL GROUP CO., LTD. (CN) 2023-08-09 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230357242-A1 COMPOUND AS AKT KINASE INHIBITOR AKT2, MTOR, AKT1 OPRD1 4575/4885L3MBTL3 4811/4885L3MBTL1 4657/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.