SCHEMBL2596691

SCHEMBL2596691

CCc1cc(-c2nnc(OC(N)=O)n2-c2cccc3[nH]c(C)cc23)c(O)cc1O

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DAO P14920 1/20 0.33
DDO Q99489 1/20 0.33
HSP90AA1 P07900 9/20 0.33
PRKCA P17252 1/20 0.32
PRKCQ Q04759 1/20 0.32
KDM4E B2RXH2 1/20 0.32
ALDH1A1 P00352 1/20 0.32
LMNA P02545 1/20 0.32
MAPT P10636 1/20 0.32
HPGD P15428 1/20 0.32
TSHR P16473 1/20 0.32
HSD17B10 Q99714 1/20 0.32
SYK P43405 3/20 0.32
GAA P10253 1/20 0.32
F2 P00734 1/20 0.31
F12 P00748 1/20 0.31
ALOX15 P16050 1/20 0.31
ALOX12 P18054 1/20 0.31
ABCB11 O95342 1/20 0.30
HTR1A P08908 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9925250 0.88 GOT1 (0.36) HSP90AA1MAPTGAA
SCHEMBL419803 0.81 HSD11B1 (0.38) HSP90AA1KDM4ELMNAMAPTGAA
SCHEMBL12180120 0.77 AOC3 (0.38) KDM4EALDH1A1LMNAMAPTHPGD
SCHEMBL3974853 0.77 ALDH1A1 (0.35) DAODDOHSP90AA1PRKCAPRKCQ
SCHEMBL806552 0.76 GAA (0.34) SYKGAA
SCHEMBL2596689 0.76 DAO (0.34) DAODDOHSP90AA1KDM4EALDH1A1
SCHEMBL12908734 0.75 PDE4D (0.37) HSP90AA1KDM4EALDH1A1LMNAMAPT
SCHEMBL931405 0.74 KMT2A (0.48) KDM4EALDH1A1LMNAMAPTHPGD
SCHEMBL1539292 0.73 HSP90AA1 (0.36) DAODDOHSP90AA1KDM4EALDH1A1
SCHEMBL12180125 0.72 GOT1 (0.39) ALDH1A1MAPTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011146801-A1 FORMULATION AND DOSING OF HSP90 INHIBITORY COMPOUNDS SYNTA PHARMACEUTICALS CORP. (US) 2011-11-24 WO claimed
WO-2011146801-A1 FORMULATION AND DOSING OF HSP90 INHIBITORY COMPOUNDS SYNTA PHARMACEUTICALS CORP. (US) 2011-11-24 WO disclosed