SCHEMBL2596689

SCHEMBL2596689

CCc1cc(-c2nnc(N)n2-c2cccc3[nH]c(C(C)C)cc23)c(O)cc1O

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DAO P14920 1/20 0.34
DDO Q99489 1/20 0.34
HSP90AA1 P07900 7/20 0.33
MAPT P10636 4/20 0.33
GAA P10253 3/20 0.33
ALDH1A1 P00352 2/20 0.33
HPGD P15428 2/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
POLB P06746 1/20 0.33
ALOX12 P18054 1/20 0.33
NPSR1 Q6W5P4 1/20 0.33
KDM4E B2RXH2 3/20 0.32
LMNA P02545 2/20 0.32
PAX8 Q06710 1/20 0.32
DHFR P00374 1/20 0.32
SLC2A1 P11166 1/20 0.32
TSHR P16473 1/20 0.31
HSD17B10 Q99714 1/20 0.31
NPEPPS P55786 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13280018 0.89 DAO (0.34) DAODDOHSP90AA1MAPTGAA
SCHEMBL1539292 0.87 HSP90AA1 (0.36) DAODDOHSP90AA1MAPTGAA
SCHEMBL930712 0.79 HCAR1 (0.37) HSP90AA1MAPTGAAALDH1A1HPGD
SCHEMBL421350 0.78 KDM4E (0.35) HSP90AA1MAPTGAAHPGDMEN1
SCHEMBL2596698 0.77 HSP90AA1 (0.41) HSP90AA1HSP90AB1
SCHEMBL2596691 0.76 DAO (0.33) DAODDOHSP90AA1MAPTGAA
SCHEMBL3974314 0.75 DAO (0.34) DAODDOHSP90AA1MAPTGAA
SCHEMBL1586624 0.74 GAA (0.33) HSP90AA1MAPTGAAALDH1A1HPGD
SCHEMBL2596685 0.73 HSP90AA1 (0.35) DAODDOHSP90AA1MAPTGAA
SCHEMBL1881956 0.71 NPEPPS (0.37) DAODDOHSP90AA1MAPTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011146801-A1 FORMULATION AND DOSING OF HSP90 INHIBITORY COMPOUNDS SYNTA PHARMACEUTICALS CORP. (US) 2011-11-24 WO disclosed