SCHEMBL25967749

SCHEMBL25967749

COC(=O)[C@@H]1CCCN1OC(=O)c1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.50
CHRNB2 P17787 1/20 0.45
CHRNA5 P30532 1/20 0.45
CHRNA7 P36544 1/20 0.45
CHRNA4 P43681 1/20 0.45
TSHR P16473 1/20 0.45
LTA4H P09960 2/20 0.45
ACE P12821 1/20 0.44
FKBP1A P62942 1/20 0.43
MEN1 O00255 1/20 0.43
ALOX5 P09917 1/20 0.42
KCNH2 Q12809 2/20 0.42
MAPT P10636 1/20 0.42
MAOA P21397 1/20 0.42
SLC6A2 P23975 1/20 0.42
SLC6A4 P31645 1/20 0.42
SCN1A P35498 1/20 0.42
SLC6A3 Q01959 1/20 0.42
SCN2A Q99250 1/20 0.42
SIGMAR1 Q99720 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20253879 0.96 KMT2A (0.46) KMT2ACHRNB2CHRNA5CHRNA7CHRNA4
SCHEMBL23746785 0.85 ALDH1A1 (0.49) KMT2ACHRNB2CHRNA5CHRNA7CHRNA4
SCHEMBL18849795 0.85 ALDH1A1 (0.49) KMT2ACHRNB2CHRNA5CHRNA7CHRNA4
SCHEMBL18474161 0.85 ALDH1A1 (0.49) KMT2ACHRNB2CHRNA5CHRNA7CHRNA4
SCHEMBL18474217 0.83 DPP4 (0.45) KMT2ACHRNB2CHRNA5CHRNA7CHRNA4
SCHEMBL18474160 0.83 DPP4 (0.45) KMT2ACHRNB2CHRNA5CHRNA7CHRNA4
SCHEMBL19099852 0.83 KMT2A (0.44) KMT2ATSHRKCNH2MAPTMAOA
SCHEMBL20253880 0.81 TDP1 (0.45) KMT2ACHRNB2CHRNA5CHRNA7CHRNA4
SCHEMBL8911799 0.80 LTA4H (0.49) KMT2ATSHRLTA4HFKBP1AALOX5
SCHEMBL7026294 0.80 LTA4H (0.49) KMT2ATSHRLTA4HFKBP1AALOX5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3810129-B1 PCSK9 ANTAGONIST BICYCLO-COMPOUNDS MERCK SHARP & DOHME LLC (US) 2023-08-16 EP disclosed