SCHEMBL2596817

SCHEMBL2596817

COc1ccc(Cc2cnc3c[nH]nc3c2I)cc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MPO P05164 1/20 0.41
POLB P06746 1/20 0.38
ALDH1A1 P00352 3/20 0.38
SMN1; SMN2 Q16637 2/20 0.38
LMNA P02545 1/20 0.38
KDM4E B2RXH2 1/20 0.37
MPI P34949 1/20 0.37
APOBEC3G Q9HC16 1/20 0.37
LTA4H P09960 1/20 0.37
APP P05067 2/20 0.37
PDGFRB P09619 1/20 0.36
PDGFRA P16234 1/20 0.36
CYP11B1 P15538 3/20 0.36
CYP11B2 P19099 3/20 0.36
VNN1 O95497 1/20 0.35
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
CNR1 P21554 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1753882 0.68 LTA4H (0.46) MPOALDH1A1SMN1; SMN2LMNAKDM4E
SCHEMBL17713797 0.68 LTA4H (0.46) MPOPOLBALDH1A1SMN1; SMN2LMNA
SCHEMBL28166476 0.66 ALDH1A1 (0.46) MPOPOLBALDH1A1SMN1; SMN2LMNA
SCHEMBL27585502 0.64 NPSR1 (0.44) POLBALDH1A1SMN1; SMN2LMNALTA4H
SCHEMBL27298346 0.64 LTA4H (0.53) MPOALDH1A1SMN1; SMN2LMNAKDM4E
SCHEMBL8376680 0.63 DHFR (0.76) LMNA
SCHEMBL28212221 0.63 SLC2A1 (0.52) MPOALDH1A1KDM4EMPIAPOBEC3G
SCHEMBL7716578 0.63 PLA2G7 (0.48) MPOPOLBALDH1A1SMN1; SMN2LMNA
SCHEMBL27884 0.63 LTA4H (0.81) ALDH1A1SMN1; SMN2LMNALTA4H
SCHEMBL25986524 0.63 LTA4H (0.81) ALDH1A1SMN1; SMN2LMNALTA4H

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011146287-A1 PYRAZOLO[4,3-B]PYRIDINE-7-AMINE INHIBITORS OF ALK5 TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2011-11-24 WO disclosed