SCHEMBL25980680

SCHEMBL25980680

COc1ccc(CNCC(Oc2c(Br)cncc2Br)C(F)(F)F)c(OC)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
APLNR P35414 1/20 0.50
HTR2A P28223 2/20 0.47
HTR2C P28335 2/20 0.47
TSHR P16473 5/20 0.41
CYP1A2 P05177 4/20 0.41
CYP3A4 P08684 4/20 0.41
CYP2D6 P10635 4/20 0.41
CYP2C19 P33261 4/20 0.41
USP2 O75604 2/20 0.41
ALOX15 P16050 2/20 0.41
KDM4C Q9H3R0 1/20 0.39
LMNA P02545 2/20 0.38
HSD17B10 Q99714 1/20 0.38
CLK4 Q9HAZ1 1/20 0.38
ALDH1A1 P00352 3/20 0.38
CYP2C9 P11712 2/20 0.38
HDAC3 O15379 1/20 0.38
HDAC1 Q13547 1/20 0.38
HDAC2 Q92769 1/20 0.38
HDAC8 Q9BY41 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL25342537 0.99 APLNR (0.49) APLNRHTR2AHTR2CTSHRCYP1A2
SCHEMBL25980752 0.88 APLNR (0.44) APLNRHTR2AHTR2CTSHRCYP1A2
Hydrochloric Acid SCHEMBL30479625 0.87 APLNR (0.44) APLNRHTR2AHTR2CTSHRCYP1A2
Hydrochloric Acid SCHEMBL25342899 0.87 APLNR (0.44) APLNRHTR2AHTR2CTSHRCYP1A2
SCHEMBL25980671 0.81 GAA (0.40) APLNRHTR2AHTR2CTSHRCYP1A2
SCHEMBL25345233 0.77 POLB (0.43) TSHRKDM4CLMNAALDH1A1
SCHEMBL25341754 0.77 APLNR (0.63) APLNRHTR2AHTR2CHDAC3HDAC1
SCHEMBL25980674 0.75 GAA (0.39) TSHRKDM4CLMNAALDH1A1
SCHEMBL783785 0.70 APLNR (1.00) APLNRHTR2AHTR2CTSHRALDH1A1
SCHEMBL15969133 0.70 APLNR (0.73) APLNRHTR2AHTR2CTSHRHDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023148501-A1 HETEROCYCLIC DERIVATIVES AS MALT1 INHIBITORS C4X DISCOVERY LIMITED (GB) 2023-08-10 WO disclosed