SCHEMBL25980752

SCHEMBL25980752

COc1ccc(CNCC(Oc2c(Br)cnc(C)c2Br)C(F)(F)F)c(OC)c1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
APLNR P35414 1/20 0.44
HTR2A P28223 2/20 0.43
HTR2C P28335 2/20 0.43
TSHR P16473 7/20 0.38
ALDH1A1 P00352 2/20 0.38
NPSR1 Q6W5P4 1/20 0.38
CYP1A2 P05177 7/20 0.37
CYP3A4 P08684 7/20 0.37
CYP2C19 P33261 7/20 0.37
CYP2D6 P10635 5/20 0.37
ALOX15 P16050 4/20 0.37
USP2 O75604 3/20 0.37
TP53 P04637 1/20 0.36
HSD17B10 Q99714 2/20 0.36
MEN1 O00255 2/20 0.36
KMT2A Q03164 2/20 0.36
LMNA P02545 1/20 0.35
CLK4 Q9HAZ1 1/20 0.35
HDAC3 O15379 1/20 0.35
HDAC1 Q13547 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL30479625 0.99 APLNR (0.44) APLNRHTR2AHTR2CTSHRALDH1A1
Hydrochloric Acid SCHEMBL25342899 0.99 APLNR (0.44) APLNRHTR2AHTR2CTSHRALDH1A1
SCHEMBL25980680 0.88 APLNR (0.50) APLNRHTR2AHTR2CTSHRALDH1A1
Hydrochloric Acid SCHEMBL25342537 0.87 APLNR (0.49) APLNRHTR2AHTR2CTSHRALDH1A1
SCHEMBL30479644 0.79 HTR2A (0.54) APLNRHTR2AHTR2CTSHRALDH1A1
SCHEMBL25343094 0.79 HTR2A (0.54) APLNRHTR2AHTR2CTSHRALDH1A1
SCHEMBL25341773 0.79 GAA (0.40) TSHRALDH1A1NPSR1MEN1KMT2A
SCHEMBL25980741 0.76 GAA (0.38) TSHRALDH1A1NPSR1MEN1KMT2A
SCHEMBL25341754 0.72 APLNR (0.63) APLNRHTR2AHTR2CMEN1KMT2A
SCHEMBL25980671 0.71 GAA (0.40) APLNRHTR2AHTR2CTSHRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023148501-A1 HETEROCYCLIC DERIVATIVES AS MALT1 INHIBITORS C4X DISCOVERY LIMITED (GB) 2023-08-10 WO disclosed