SCHEMBL2598936

SCHEMBL2598936

CCCCCC(=O)OCOP(=O)(O)C(O)(CCCN)P(=O)(OCOC(=O)CCCCC)OCOC(=O)CCCCC

nearest known ligand 0.40

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ENPP2 Q13822 6/20 0.40
LPAR3 Q9UBY5 4/20 0.40
LPAR1 Q92633 3/20 0.40
LPAR6 P43657 1/20 0.40
LPAR4 Q99677 1/20 0.40
LPAR5 Q9H1C0 1/20 0.40
LPAR2 Q9HBW0 1/20 0.40
FDPS P14324 7/20 0.40
PDE3A Q14432 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.39
GGPS1 O95749 3/20 0.39
DGKA P23743 1/20 0.39
CYP1A2 P05177 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2599116 0.94 ENPP2 (0.43) ENPP2LPAR3LPAR1LPAR6LPAR4
SCHEMBL9500079 0.84 ENPP2 (0.41) ENPP2LPAR3LPAR1LPAR6LPAR4
SCHEMBL2453742 0.81 FDPS (0.41) FDPSPDE3AGGPS1CYP1A2
SCHEMBL2458967 0.81 FDPS (0.42) FDPSPDE3A
SCHEMBL2455650 0.81 FDPS (0.42) FDPSPDE3A
SCHEMBL2463502 0.80 FDPS (0.40) FDPSPDE3A
SCHEMBL9188504 0.80 FDPS (0.41) FDPSPDE3A
SCHEMBL9190696 0.75 HTT (0.46) SMN1; SMN2
SCHEMBL2598916 0.73 FDPS (0.46) FDPSPDE3AGGPS1
SCHEMBL5995956 0.72 FDPS (0.37) FDPSPDE3ACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0416689-B1 Acyloxymethyl esters of bisphosphonic acids as bone resorption inhibitors MERCK & CO INC (US) 1995-11-29 EP claimed
US-5227506-A Acyloxymethyl esters of bisphosphonic acids as bone resorption inhibitors MERCK & CO., INC. (US) 1993-07-13 US claimed
WO-2011146819-A2 METHODS AND COMPOSITIONS FOR TREATMENT NF-κB-MEDIATED AND α7 INTEGRIN-SUPPRESSED DISEASES DMD THERAPIES, LLC (US) 2011-11-24 WO disclosed
EP-0416689-B1 Acyloxymethyl esters of bisphosphonic acids as bone resorption inhibitors MERCK & CO INC (US) 1995-11-29 EP disclosed
US-5227506-A Acyloxymethyl esters of bisphosphonic acids as bone resorption inhibitors MERCK & CO., INC. (US) 1993-07-13 US disclosed
EP-0416689-A2 Acyloxymethyl esters of bisphosphonic acids as bone resorption inhibitors MERCK & CO. INC. (US) 1991-03-13 EP disclosed